机译:趋化因子受体CXCR4蛋白接口的基于结构的配体发现
Department of Pharmaceutical Chemistry, University of California, San Francisco, CA 94158;
Department of Pharmaceutical Chemistry, University of California, San Francisco, CA 94158;
Department of Biochemistry, Medical College of Wisconsin, Milwaukee, WI 53226;
Centre de Recherche, Centre Hospitalier Universitaire Sainte-Justine, Montreal, QC, Canada H3T 1C5,Department of Biochemistry, Universite de Montreal, Montreal, QC, Canada H3T 1J4;
Department of Pharmaceutical Chemistry, University of California, San Francisco, CA 94158;
Department of Pharmaceutical Chemistry, University of California, San Francisco, CA 94158;
Centre de Recherche, Centre Hospitalier Universitaire Sainte-Justine, Montreal, QC, Canada H3T 1C5,Department of Biochemistry, Universite de Montreal, Montreal, QC, Canada H3T 1J4;
Department of Pharmaceutical Chemistry, University of California, San Francisco, CA 94158;
Department of Biochemistry, Medical College of Wisconsin, Milwaukee, WI 53226;
drug design; virtual screening; promiscuous aggregation;
机译:肝素寡糖抑制趋化因子(CXC基序)配体12(CXCL12)心脏保护,通过与二聚化界面结合,促进低聚,并与趋化因子(CXC基序)受体4(CXCR4)N末端竞争
机译:半胱氨酸-X-半胱氨酸基质趋化因子配体12及其受体CXCR4:在猪早期妊娠期间母体概念界面的表达,调节和可能的功能
机译:基于结构配体的新型配体靶向趋化因子-G-蛋白质-偶联受体界面内的多个位点
机译:通过利用多脯氨酸螺旋作为接头,通过利用多脯氨酸螺旋进行趋化因子受体CXCR4的二价配体
机译:阐明趋化因子CXCL12及其受体CXCR4和CXCR7在癌症中的功能和信号传导机制。
机译:基于结构的配体发现趋化因子受体CXCR4的蛋白-蛋白界面
机译:基于结构的配体发现趋化因子受体CXCR4的蛋白-蛋白界面