首页> 外国专利> AGENT FOR INHIBITING REDUCTION OF DECOMPOSITION OF MODIFIED ELASTIN, AGENT FOR MAINTAINING NORMAL ELASTIC FIBERS, AGENT FOR INHIBITING FORMATION OF ELASTIN-ELAFIN COMPLEX, AND COMPOSITION CONTAINING SAID AGENTS

AGENT FOR INHIBITING REDUCTION OF DECOMPOSITION OF MODIFIED ELASTIN, AGENT FOR MAINTAINING NORMAL ELASTIC FIBERS, AGENT FOR INHIBITING FORMATION OF ELASTIN-ELAFIN COMPLEX, AND COMPOSITION CONTAINING SAID AGENTS

机译:用于抑制改性弹性蛋白的分解的药剂,用于保持正常弹性纤维的药剂,用于抑制Elastin-Elafin络合物的形成的试剂,以及含有所述药剂的组合物

摘要

The purpose of the present invention is to provide an agent for inhibiting formation of an elastin-elafin complex and a composition for inhibiting formation of an elastin-elafin complex, the agent and composition being capable of inhibiting formation of an elastin-elafin complex. The present invention pertains to an agent for inhibiting reduction of decomposition of modified elastin, the agent containing, as an active ingredient, a compound represented by general formula (I) and/or a derivative thereof. (In formula (I), R1-R4 may be the same or different and represent a hydrogen atom or a hydroxy group. When R1 is a hydrogen atom, R2 is a hydroxy group. When R1 is a hydroxy group, R2 is a hydrogen atom. When R3 is a hydrogen atom, R4 is a hydroxy group. When R3 is a hydroxy group, R4 is a hydrogen atom.)
机译:本发明的目的是提供一种用于抑制ELASTIN-ELAFIN复合物的形成的试剂,以及用于抑制弹性蛋白 - ELAFIN络合物的形成,药剂和组合物能够抑制ELASTIN-ELAFIN复合物的形成。 本发明涉及用于抑制改性弹性蛋白的分解的药剂,含有含有活性成分的试剂,其由通式(I)和/或其衍生物表示的化合物。 (在式(I)中,R1-R4可以相同或不同,代表氢原子或羟基。当R1是氢原子时,R 2是羟基。当R1是羟基时,R 2是氢气 原子。当R3是氢原子时,R 4是羟基。当R3是羟基时,R 4是氢原子。)

著录项

  • 公开/公告号WO2021200705A1

    专利类型

  • 公开/公告日2021-10-07

    原文格式PDF

  • 申请/专利权人 SUNTORY HOLDINGS LIMITED;

    申请/专利号WO2021JP13020

  • 发明设计人 AKAZAWA SOTA;KITAGAWA SAYURI;

    申请日2021-03-26

  • 分类号A61K31/7004;A61P17;A61P43;

  • 国家 JP

  • 入库时间 2022-08-24 21:33:34

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