Acryloyl-piperazines of formula (I) and their acid addn. salts. (where R is lower alkyl; R1 and R2 are lower alkyl, or H (with the condition that both cannot be H); and R3 is H or lower alkyl) are anaesthetics. Cpd. KA-100 is an anaesthetic, which shows anti-nociceptive activity and has good analgesic and muscle relaxant activity.
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机译:式(I)的丙烯酰基-哌嗪及其酸加成。盐。 (其中R为低级烷基; R 1和R 2为低级烷基,或H(在不能都为H的条件下;并且R 3为H或低级烷基)是麻醉剂。 CPD。 KA-100是麻醉剂,具有抗伤害感受活性,并具有良好的止痛和肌肉松弛作用。
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