An oxazoline deriv. of formula (I) is prepd. by reacting compds. of formula (II) with compds. of formula (III) in an inactive organic solvent, then applying ultraviolet rays. In the formulas, R1 and R2 are H, halogen, or lower alkyl; R3,R4,R5,R6 and R7 are H or lower alkyl; and R8 is H, lower alkyl, or formyl. (I) is an orally active antidiabetic agent.
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机译:恶唑啉衍生物。制备式(I)的化合物。通过反应compds。式(II)的化合物。式(III)的化合物在惰性有机溶剂中,然后施加紫外线。式中,R 1和R 2为H,卤素或低级烷基。 R3,R4,R5,R6和R7为H或低级烷基; R 8为H,低级烷基或甲酰基。 (I)是口服活性抗糖尿病药。
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