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A process for the preparation of New Antibiotics, especially derived from UNWTO, modified in C - 23.
A process for the preparation of New Antibiotics, especially derived from UNWTO, modified in C - 23.
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机译:一种新抗生素的制备方法,特别是从世贸组织衍生的新抗生素,经C-23修饰。
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摘要
Process for the preparation of New Antibiotics, especially derived from UNWTO modified C - 23.Consists of: (a) submit a compound of formula (i), where r is an azido Reduction reaction with triphenylphosphine to a temperature of between 0 and 100jc, to form a compound of formula (i), where r is - NH2; and b) optionally, acilar amino derivative to form a compound of formula (i) Where R IS - NHR, R is an acyl Group; R IS h, alcanoilo C 1 to 5, Benzoyl and others; R IS h,Alcanoilo C 1 to 5, phenylacetylene and others; R IS h, alcanoilo C 1 to 5 and others; and R IS h, alkyl Cyclohexyl C 1 to 6, and others.
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机译:制备新抗生素的方法,尤其是从世贸组织经修饰的C-23衍生的新抗生素,包括:(a)提交式(i)的化合物,其中r为与三苯膦的叠氮基还原反应,温度为0至100jc,形成式(i)的化合物,其中r为-NH 2; b)任选地,氨基芳基衍生物形成式(i)的化合物,其中R是-NHR,R是酰基; R IS h,Alcanoilo C 1至5,苯甲酰基等; R IS h,Alcanoilo C 1至5,苯乙炔等; R IS h,阿尔卡诺伊洛C 1至5等; R 1为烷基,环己基C 1至6等。
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