首页> 外国专利> COMPOUNDS HAVING A COGNITION ADJUVANT ACTON AGENTS CONTAINING THEM,AND THE USE THERE OF THE TREATMENT AND PROPHYLAXIS OF COGNITIVES DYSFUNCTIONS

COMPOUNDS HAVING A COGNITION ADJUVANT ACTON AGENTS CONTAINING THEM,AND THE USE THERE OF THE TREATMENT AND PROPHYLAXIS OF COGNITIVES DYSFUNCTIONS

机译:具有包含它们的认知助剂的化合物,以及治疗认知功能障碍的前瞻性药物

摘要

The compounds (I) having a cognition adjuvant action and agants containing them are prepared. In (I), n is 1 or 2; R is hydrogen, C1- C18 alkyl, CaH(2a-b+1) aliphatic acyclic radical, or CcH(2c-d-1) mono-, di-, tri-, and tetra-, etc.; R1 is hydrogen, C1-C18 alkyl, CaH(2a-b+1) acyclic aliphatic radical or CcH(2c-d-1) mono-, di-, t6ri- and tetraa-, etc.; R2 and R3 are equal, hydrogen, di(C1-C4)- alkylamino-(C1-C5)-aroyloxy-(C1-C8) alkyl or (C1-C6)- alkoxycarbonyloxy-(C1-C6)-alkyl etc.; R4 and R5 are cyclic ring systems having mono-, di- or tricyclic hetero cyclic ring.
机译:制备具有认知佐剂作用的化合物(I)和包含它们的助剂。在(I)中,n为1或2; R为氢,C1-C18烷基,CaH(2a-b + 1)脂族无环基团或CcH(2c-d-1)单,二,三和四等; R1是氢,C1-C18烷基,CaH(2a-b + 1)无环脂族基团或CcH(2c-d-1)单,二,t6ri-和tetraa-等; R2和R3相同,为氢,二(C1-C4)-烷基氨基-(C1-C5)-芳氧基-(C1-C8)烷基或(C1-C6)-烷氧基羰氧基-(C1-C6)-烷基等。 R4和R5是具有单,二或三环杂环的环系统。

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