首页> 外国专利> SALTS OF MESIDIDES OF ALPHA-PIPERIDINCARBOXYLIC ACIDS POSSESSING LOCALLYANESTHETIC, ANTIARYTHMIC AND ANTIFIBRILLATORY ACTIVITY AND MESIDIDES OF ALPHA-PUPERIDINCARBOXYLIC ACIDS AS INTERMEDIATE PRODUCTS FOR SYNTHESIS OF SALTS OF MESIDIDES OF PIPERIDINCARBOXYLIC ACIDS

SALTS OF MESIDIDES OF ALPHA-PIPERIDINCARBOXYLIC ACIDS POSSESSING LOCALLYANESTHETIC, ANTIARYTHMIC AND ANTIFIBRILLATORY ACTIVITY AND MESIDIDES OF ALPHA-PUPERIDINCARBOXYLIC ACIDS AS INTERMEDIATE PRODUCTS FOR SYNTHESIS OF SALTS OF MESIDIDES OF PIPERIDINCARBOXYLIC ACIDS

机译:具有局部麻醉,抗炎和抗纤维化活性的α-哌啶羧酸的半胱氨酸盐和α-泛脂酰羧胺的中间体

摘要

1. salt.u043cu0435u0437u0438u0434u0438u0434u043eu0432 - u043fu0438u043fu0435u0440u0438u0434u0438u043du043au0430u0440u0431u043eu043du043eu0432u044bu0445 acids common formula and sn - them CONH - n i r where r - n - butyl or u0438u0437u043eu0431u0443u0442u0438u043b; x is chlorine or bromine, with u043cu0435u0441u0442u043du043eu0430u043du0435u0441u0442u0435u0437u0438u0440u0443u044eu0449u0435u0439, u0430u043du0442u0438u0430u0440u0438u0442u043c u0438u0447u0435u0441u043au043eu0439 and u0430u043du0442u0438u0444u0438u0431u0440u0438u043bu043bu00a0u0442u043eu0440u043du043eu0439 activity. 2. u043cu0435u0437u0438u0434u0438u0434u044b o.- u043fu0438u043fu0435u0440u0438u0434u0438u043du043au0430u0440u0431u043eu043du043eu0432u044bu0445 acids of general formula cl to) CONH trademark) r r sp where r n butyl or u0438u0437u043eu0431u0443u0442u0438u043b, 4 as intermediate products u0434u043bu00a0 synthesis of salts u043cu0435u0437u0438u0434u0438u0434u043eu0432 u043e6 - u043fu0438u043fu0435u0440u0438u0434u0438 u043du043au0430u0440u0431u043eu043du043eu0432u044bu0445 acids.
机译:1.盐。 u043c u0435 u0437 u0438 u0434 u0438 u0434 u043e u0432- u043f u0438 u043f u0435 u0440 u0438 u0434 u0438 u043d u043d u043a u0430 u0440 u0431 u043e u043d u043e u0432 u044b u0445酸的通用配方和sn-它们是CONH-nir,其中r-n-丁基或 u0438 u0437 u043e u043e u0431 u0443 u0442 u0438 u043b; x是氯或溴,具有 u043c u0435 u0441 u0442 u043d u043e u0430 u043d u0435 u0441 u0442 u0435 u0437 u0438 u0440 u0443 u0443 u044e u0449 u0435 u0439, u0430 u043d u0442 u0438 u0430 u0440 u0438 u0442 u043c u0438 u0447 u0435 u0441 u043a u043e u0439和 u0430 u043d u0442 u0438 u0444 u0438 u0431 u0440 u0440 u0 u043b u043b u00a0 u0442 u043e u0440 u043d u043e u0439活动。 2. u043c u0435 u0437 u0438 u0434 u0438 u0434 u044b o。- u043f u0438 u043f u0435 u0440 u0438 u0434 u0438 u043d u043d u043a u0430 u0440 u0431 u043e u043d u043e u0432 u044b u0445带有CONH商标的酸)rr sp其中rn丁基或 u0438 u0437 u043e u0431 u0443 u0442 u0438 u043b,4作为中间产物 u0434 u043b u00a0盐的合成 u043c u0435 u0437 u0438 u0434 u0438 u0434 u043e u0432 u043e6- u043f u0438 u043f u0435 u0440 u0438 u0434 u0438 u043d u043a u0430 04 u0431 u043e u043d u043e u0432 u044b u0445酸。

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