首页> 外国专利> CRYSTALLINE FORMS OF ENDO-2,3-DIHYDRO-N- £8-METHYL-8-AZABICYCLO(3,2,1)OCT-3-YL -2-OXO-1H-BENZIMIDAZOLE-1-CARBOXAMIDE HYDROCHLORIDE MONOHYDRATE, ENDO-3-ETHYL-2,3-DIHYDRO- ... HYDROCHLORIDE AMMONIUM HYDRATE

CRYSTALLINE FORMS OF ENDO-2,3-DIHYDRO-N- £8-METHYL-8-AZABICYCLO(3,2,1)OCT-3-YL -2-OXO-1H-BENZIMIDAZOLE-1-CARBOXAMIDE HYDROCHLORIDE MONOHYDRATE, ENDO-3-ETHYL-2,3-DIHYDRO- ... HYDROCHLORIDE AMMONIUM HYDRATE

机译:ENDO-2,3-二氢-N-£8-甲基-8-氮杂双(3,2,1)OCT-3-YL的结晶形式| -2-氧代-1H-苯并咪唑-1-碳酰氢一一水合物,内酯-3-乙基-2,3-二氢-...氢氧一酸一铵

摘要

In the present invention there is disclosed a crystalline monohydrate of endo-2,3-dihydro-N-(8-methyl-8-azabicyclo[3,2,1]oct-3-yl)-2-oxo-1H-benzimidazole-1-carboxamide hydrochloride of the general formula 2a in which R represents a hydrogen atom. In the present invention there are also claimed processes for its preparation as well as pharmaceutical preparations in which said compound is comprised.
机译:在本发明中,公开了内-2,3-二氢-N-(8-甲基-8-氮杂双环[3,2,1]辛-3-基)-2-氧代-1H-苯并咪唑的结晶一水合物通式2a的-1-甲酰胺盐酸盐,其中R表示氢原子。在本发明中,还要求保护其制备方法以及包含所述化合物的药物制剂。

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