首页> 外国专利> PROCESS FOR PREPARING ISOMERS, OR PHARMACEUTICALLY ACCEPTABLE SALTS, AND ALDEHYDE AS AN INTERMEDIATE PRODUCT IN THE 1-ALKYL, 1-ALKENYL OR 1-ALKYNYLARYL-2-AMINO-1, 3- PROPANEDIOL SYSTEM

PROCESS FOR PREPARING ISOMERS, OR PHARMACEUTICALLY ACCEPTABLE SALTS, AND ALDEHYDE AS AN INTERMEDIATE PRODUCT IN THE 1-ALKYL, 1-ALKENYL OR 1-ALKYNYLARYL-2-AMINO-1, 3- PROPANEDIOL SYSTEM

机译:在1-烷基,1-烯基或1-炔基-2-氨基-1,3-丙烷体系中制备中间体的异构体或药学上可接受的盐和醛的方法

摘要

FIELD: used as antiphlogistics. SUBSTANCE: in order to prepare 1-alkynylpyridinyl-2- amino-1, 3-propanediol, pyridinylcarboxaldehyde is condensed with amidomalonic acid ester, followed, if necessary, by hydrogenation or hydrolysis of the resulting product. EFFECT: improved properties of the resulting product. 3 cl
机译:领域:用作消炎药。物质:为了制备1-炔基吡啶基-2-氨基-1,3-丙二醇,将吡啶基甲醛与酰胺基丙二酸酯缩合,然后,如果需要,将所得产物氢化或水解。效果:改善了所得产品的性能。 3厘升

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