首页> 外国专利> BRADYARRHYTHMIA TREATING AGENT

BRADYARRHYTHMIA TREATING AGENT

机译:缓慢型心律失常治疗剂

摘要

PURPOSE: To obtain the subject treating agent containing a carbostyril derivative having a specific structure as an active ingredient, exhibiting remarkable action, especially on sick sinus syndrome, useful also for complication of intraatrial thrombus due to bradyarrhythmia and free from adverse effect. ;CONSTITUTION: This treating agent contains a compound of the formula (A is a lower alkylene; R is a cycloalkyl; the bond between 3 and 4 positions of carbostyril skeleton is single bond or double bond) or its salt, preferably 6-[4-(1- cyclohexyl-1,2,3,4-tetrazol-5-yl)butoxy]-3,4-dihydrocarbostyril or its salt as an active ingredient. The content of the compound of the compound is preferably 5-50wt.% per total composition. The daily dose of the compound of the formula is normally preferably 0.6-50mg/kg.weight. The compound of the formula contains preferably 10-1000mg active ingredient in the administration unit form.;COPYRIGHT: (C)1996,JPO
机译:用途:获得包含具有特定结构的咔唑衍生物作为活性成分的主题治疗剂,该治疗剂表现出显着的作用,特别是对病态窦房结综合症,也可用于由于心律失常引起的房内血栓并发症并且没有不良作用。 ;组成:该处理剂含有下式的化合物或其盐,优选为6- [4]:A为低级亚烷基; R为环烷基; Carbostyril骨架的3至4位之间的键为单键或双键) -(1-环己基-1,2,3,4-四唑-5-基)丁氧基] -3,4-二烃基丁酮或其盐作为有效成分。化合物中化合物的含量相对于全部组合物优选为5〜50重量%。式的化合物的日剂量通常优选为0.6-50mg / kg。体重。该式的化合物优选以给药单位形式包含10-1000mg的活性成分。;版权所有:(C)1996,JPO

著录项

  • 公开/公告号JPH08268891A

    专利类型

  • 公开/公告日1996-10-15

    原文格式PDF

  • 申请/专利权人 OTSUKA PHARMACEUT CO LTD;

    申请/专利号JP19950072985

  • 发明设计人 SHIN HIROTSUGU;SAITO HIROKAZU;

    申请日1995-03-30

  • 分类号A61K31/47;

  • 国家 JP

  • 入库时间 2022-08-22 04:03:48

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号