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USE OF NATURAL CYCLODEXTRINES AND THEIR DERIVATIVES FOR SOLUBILIZING MATERIALS OF TROMBOCITE-AGGREGATION-INHIBITING ACTIVITY IN THE GINKGOLIDE'S FAMILY
USE OF NATURAL CYCLODEXTRINES AND THEIR DERIVATIVES FOR SOLUBILIZING MATERIALS OF TROMBOCITE-AGGREGATION-INHIBITING ACTIVITY IN THE GINKGOLIDE'S FAMILY
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机译:天然环糊精及其衍生物在银杏内酯家族中的锂辉石聚集抑制活性增溶中的应用
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摘要
Solubilising a ginkgolide platelet-activating factor antagonist (I) in aq. media comprises combining (I) with a cyclodextrin of formula (II) to form a water-soluble clathrate: n = 6-8; R1 = OH or SR2, and R2 = a gp. derived from a mono- or oligosaccharide. Also claimed are clathrates as above.
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