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HIGH AFFINITY, BENZYLPIPERIDINE DERIVATIVES TO BINDING POINTS OF AMINO ACID RECEPTORS
HIGH AFFINITY, BENZYLPIPERIDINE DERIVATIVES TO BINDING POINTS OF AMINO ACID RECEPTORS
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机译：高亲和力，苄基哌啶衍生物对氨基酸受体的结合点
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摘要
Benzyl substd. piperidinoalkyl heterobicyclyl ketones and alcohols and their salts are new: R1 = H; halo; or NO2; R2 = 2-, 3- or 4-benzyl opt. ring substd. by halo; R3 = H or A; A = 1-6C alkyl; B = O or (H)(OH); halo = F, Cl, Br or I; n = 0-2; X = CO or SO2; Y = CH2; NH; O; S; or CO when X = CO and Z = NH or NA; and Z = CH2; C(A)2; CH2-CH2; CH=CH; CO; NH; O; or a bond; and 1 of X, Y and Z can be O, S or NH; cpds. are excluded when R2 = 4-benzyl, X = CO, Y = Z = CH2 and R1=H; and when X-Y or Y-Z = -O-O-, -S-S-, -NH-O-, -O-NH-, -NH-NH-, -O-S- or -S-O.
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机译：苄基取代。哌啶子基烷基杂双环基酮和醇及其盐是新的：R 1 ＝ H;光环;或NO2; R 2 ＝ 2-，3-或4-苄基。环取代。晕R 3 ＝ H或A; A = 1-6C烷基; B = O或（H）（OH）;卤素= F，Cl，Br或I; n = 0-2; X = CO或SO2; Y = CH2; NH; O; S;当X = CO且Z = NH或NA时为CO; Z = CH2; C（A）2; CH2-CH2; CH = CH;一氧化碳NH; O;或债券; X，Y和Z中的1个可以是O，S或NH; cpds。当R 2 ＝ 4-苄基，X ＝ CO，Y ＝ Z ＝ CH 2且R 1 ＝ H时，排除在外;当X-Y或Y-Z = -O-O-，-S-S-，-NH-O-，-O-NH-，-NH-NH-，-O-S-或-S-O时。
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