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SYNTHETIC EXCITATORY AMINO ACIDS, PREPARATION METHOD THEREOF, INTERMEDIATES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

机译:合成兴奋性氨基酸,其制备方法,其制备中间体和包含相同成分的药物组合物

摘要

Compounds of Formula (I) wherein X is (CH 2) n wherein n is 1; R 2 is CO 2 R 4 and R 3 is hydrogen or R 2 is hydrogen and R 3 is CO 2 R 4; R 1 and R 4 are independently hydrogen, C 1-10 alkyl, C 2-10 alkenyl, aryl or arylalkyl, or a pharmaceutically acceptable salt thereof; how to prepare them; an intermediate for their preparation and a pharmaceutical composition containing the same
机译:式(I)的化合物,其中X为(CH 2)n其中n为1; R 2为CO 2 R 4且R 3为氢或R 2为氢且R 3为CO 2 R 4; R 1和R 4独立地是氢,C 1-10烷基,C 2-10烯基,芳基或芳基烷基或其药学上可接受的盐;如何准备它们;用于其制备的中间体和包含该中间体的药物组合物

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