首页> 外国专利> LINEAR POLYAMINS REPLACED WITH PIPERIDINIL-2-RENT FOR THE REDUCTION OF LEVELS OF INTRACELLULAR ENDOGEN POLYAMINS, SUCH AS PUTRESCINE, Spermidine and Spermine, and their impact on cell profiling.

LINEAR POLYAMINS REPLACED WITH PIPERIDINIL-2-RENT FOR THE REDUCTION OF LEVELS OF INTRACELLULAR ENDOGEN POLYAMINS, SUCH AS PUTRESCINE, Spermidine and Spermine, and their impact on cell profiling.

机译:取代哌替尼-2-租金的线性多胺,用于减少细胞内内源多聚糖的水平,如PUTRESCINE,亚精胺和亚精胺,及其对细胞谱分析的影响。

摘要

THE INVENTION IS ABOUT FORMULA COMPOUNDS (I), IN WHICH R {SUB, 1} IS HYDROGEN AND R {SUB, 2} IT IS LOWER RENT, LOWER RENT OR LOWER RENT, M IS 3 OR 4, AND N IS 2 OR 3; OR R {SUB, 1} AND R {SUB, 2} TOGETHER ARE TETRAMETILENE, M IS 3 OR 4, AND N IS 2; OR SALTS OF THE SAME. THE FORMULA COMPOUNDS (I) INFLUENCE IN THE POLYAMINE BIOSYNTHESIS, AND HAVE ANTIPROLIFERATIVE ACTIVITY AND ALSO ACT AGAINST PROTOZOOS.
机译:本发明是关于式(I)的化合物,其中R {SUB,1}是氢,R {SUB,2}是低价,低价或低价,M为3或4,N为2或3 ;或R {SUB,1}和R {SUB,2}一起为四金属烯,M为3或4,N为2;或相同的盐。式(I)对多胺生物合成的影响,并且具有抗增殖活性并且还对原生动物起作用。

著录项

  • 公开/公告号ES2164875T3

    专利类型

  • 公开/公告日2002-03-01

    原文格式PDF

  • 申请/专利权人 NOVARTIS AG;

    申请/专利号ES19960906733T

  • 发明设计人 FREI JORG;STANEK JAROSLAV;

    申请日1996-03-04

  • 分类号C07D211/26;A61K31/445;

  • 国家 ES

  • 入库时间 2022-08-22 00:41:36

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