首页> 外国专利> METHOD FOR TESTING THE INHIBITING ACTIVITY OF A COMPOUND ON AN ENZYME OR FOR TESTING THE RESISTANCE OF AN ENZYME AGAINST INHIBITING ACTIVITY OF A COMPOUND

METHOD FOR TESTING THE INHIBITING ACTIVITY OF A COMPOUND ON AN ENZYME OR FOR TESTING THE RESISTANCE OF AN ENZYME AGAINST INHIBITING ACTIVITY OF A COMPOUND

机译:测试化合物在酶上的抑制活性或测试酶对化合物的抑制活性的方法

摘要

The invention relates to the detection or diagnosis of genetically based enzymatic activity and/or resistance to enzyme inhibitors. The invention provides a method using an enzyme-based assay which is faster, less expensive and less facility-dependent than currently available methods for measuring the resistance to enzyme inhibitors are. The invention provides for testing the inhibiting activity of a compound on an enzyme, or the resistance of said enzyme against said inhibiting activity.
机译:本发明涉及检测或诊断基于遗传的酶活性和/或对酶抑制剂的抗性。本发明提供了一种使用基于酶的测定的方法,该方法比目前可获得的用于测量对酶抑制剂的抗性的方法更快,更便宜,且设施依赖性更低。本发明用于测试化合物对酶的抑制活性,或所述酶对所述抑制活性的抗性。

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