首页> 外国专利> Process for the simple preparation of (3-chloro-4-fluorophenyl) - 7 (3-morpholin-4-yl-propoxy) -6-ni troquinazolin-4-yl amine or (3-chloro-4-fluorophenyl) - 7- (3-morpholin-4-yl-propoxy) -6-a minoquinazolin-4-yl -amine

Process for the simple preparation of (3-chloro-4-fluorophenyl) - 7 (3-morpholin-4-yl-propoxy) -6-ni troquinazolin-4-yl amine or (3-chloro-4-fluorophenyl) - 7- (3-morpholin-4-yl-propoxy) -6-a minoquinazolin-4-yl -amine

机译:简单制备(3-氯-4-氟苯基)-[7(3-吗啉-4-基-丙氧基)-6-ni对喹唑啉-4-基]胺或(3-氯-4-氟苯基)的方法-[7-(3-吗啉-4-基-丙氧基)-6-氨基喹唑啉-4-基]-胺

摘要

"PROCESS FOR THE SIMPLE PREPARATION OF (3-CHLORINE-4-FLUOROFENYL) - [7- (3-MORFOLIN-4-IL-PROPoxy) -6-N ITROQUINAZOLIN-4-IL] AMINE OR (3-CHLORINE-4- FLUOROFENIL) - [7- (3-MORFOLIN-4-IL-PROPoxy) -6-A MINOQUINAZOLIN-4-IL] -AMINE ". The invention relates to a single vessel reaction for the preparation of (3-chloro-4-fluorophenyl) - [7- (3-morpholin-4-yl-propoxy) -6-nitroquinazolin-4-yl] amine ( I) or (3-chloro-4-fluorophenyl) - [7- (3-morpholino-4-yl-propoxy) -6-aminoquinazolin-4-yl] amine (VII)
机译:“简单地制备(3-氯-4-氟代烯基)-[7-(3-甲氧基4--4-丙氧基)-6-N异喹唑啉-4-IL]胺或(3-氯-4-)的方法氟苯腈)-[7-(3-甲氧苄氨-4-IL-丙氧基)-6-氨基喹唑啉-4-IL]-胺。本发明涉及用于制备(3-氯-4-氟苯基)-[7-(3-吗啉-4-基-丙氧基)-6-硝基喹唑啉-4-基]胺的单容器反应(I)或(3-氯-4-氟苯基)-[7-(3-吗啉代-4-基-丙氧基)-6-氨基喹唑啉-4-基]胺(VII)

著录项

  • 公开/公告号BR0108695A

    专利类型

  • 公开/公告日2002-12-10

    原文格式PDF

  • 申请/专利权人 GOEDECKE GMBH;

    申请/专利号BR20010108695

  • 申请日2001-01-23

  • 分类号C07D239/94;

  • 国家 BR

  • 入库时间 2022-08-22 00:03:50

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号