首页> 外国专利> (3-Chloro-4-fluorophenyl)-7- (3-morpholin-4-yl-propoxy) -6-nitroquinazolin-4-yl -amine or (3-chloro-4-fluorophenyl)- Simple process for the preparation of 7- (3-morpholin-4-yl-propoxy) -6-aminoquinazolin-4-yl -amine

(3-Chloro-4-fluorophenyl)-7- (3-morpholin-4-yl-propoxy) -6-nitroquinazolin-4-yl -amine or (3-chloro-4-fluorophenyl)- Simple process for the preparation of 7- (3-morpholin-4-yl-propoxy) -6-aminoquinazolin-4-yl -amine

机译:(3-氯-4-氟苯基)-[7-(3-吗啉-4-基-丙氧基)-6-硝基喹唑啉-4-基]-胺或(3-氯-4-氟苯基)-[ -(3-吗啉-4-基-丙氧基)-6-氨基喹唑啉-4-基]-胺的制备

摘要

The invention concerns a one-pot reaction for the preparation of (3-chloro-4-fluorophenyl)-[7-(3-morpholin-4-yl-propoxy)-6-nitroquinazolin-4-yl]-amine (I) or of (3-chloro-4-fluorophenyl)-[7-(3-morpholino-4-yl-propoxy)-6-aminoquinazolin-4-yl]-amine (VII)
机译:本发明涉及用于制备(3-氯-4-氟苯基)-[7-(3-吗啉-4-基-丙氧基)-6-硝基喹唑啉-4-基]-胺的一锅法反应(I)或(3-氯-4-氟苯基)-[7-(3-吗啉代-4-基-丙氧基)-6-氨基喹唑啉-4-基]-胺(VII)

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