首页> 外国专利> 8-{4-3-(5-FLUORO-1??-INDOL-3-YL)PROPYL-PIPERAZINE-1-YL}-2-METHYL-4??-BENZO1,4OXAZINE-3-??N MESYLATE WITH A HIGH AFFINITY TO RECEPTOR OF DOPAMINE D2 AND SITE OF REPETITIVE ASSIMILATION OF SEROTONIN, A PHARMACEUTICAL COMPOSITION AND A METHOD FOR THE TREATMENT OF CNS DISORDERS

8-{4-3-(5-FLUORO-1??-INDOL-3-YL)PROPYL-PIPERAZINE-1-YL}-2-METHYL-4??-BENZO1,4OXAZINE-3-??N MESYLATE WITH A HIGH AFFINITY TO RECEPTOR OF DOPAMINE D2 AND SITE OF REPETITIVE ASSIMILATION OF SEROTONIN, A PHARMACEUTICAL COMPOSITION AND A METHOD FOR THE TREATMENT OF CNS DISORDERS

机译:8- {4- [3-(5-FLUORO-1α-INDOL-3-YL)丙基]-哌嗪-1-基} -2-甲基-4α-苯并[1,4]恶嗪-3 -多巴胺D 2受体亲和力高的羟甲基磺酸盐和5-羟色胺的重复同化位点,药物组合物和CNs疾病的治疗方法

摘要

The invention relates to the novel mesylate of a phenylpiperazine derivative of the formula (??). This salt has favourable properties as compared with the free base of this compound. (??)
机译:本发明涉及式(β)的苯基哌嗪衍生物的新型甲磺酸酯。与该化合物的游离碱相比,该盐具有有利的性质。 (??)

著录项

  • 公开/公告号UA74055C2

    专利类型

  • 公开/公告日2003-10-15

    原文格式PDF

  • 申请/专利权人

    申请/专利号UA20030098662

  • 发明设计人

    申请日2002-02-19

  • 分类号C07D413/12;A61K31/538;A61P25/00;C07D265/36;

  • 国家 UA

  • 入库时间 2022-08-22 00:01:08

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