首页> 外国专利> METHOD FOR TREATMENT AND PREVENTION OF DISTURBANCES OF THE CENTRAL NERVOUS SYSTEM ASSOCIATED WITH AN ALTERATION OF GLUTAMATERGIC NEUROTRANSMISSION BY ADMINISTRATION OF 2-AMINOBENZENESULFONAMIDE DERIVATIVES

METHOD FOR TREATMENT AND PREVENTION OF DISTURBANCES OF THE CENTRAL NERVOUS SYSTEM ASSOCIATED WITH AN ALTERATION OF GLUTAMATERGIC NEUROTRANSMISSION BY ADMINISTRATION OF 2-AMINOBENZENESULFONAMIDE DERIVATIVES

机译:通过管理2-氨基苯甲磺酰胺衍生物改变和调节谷氨酸神经发射而引起的中枢神经系统疾病的治疗和预防方法

摘要

2-aminobenzenesulfonamide derivatives are used for the treatment or prevention of the disturbances of the central nervous system associated with a positive or negative modulation of glutamatergic neurotransmission, such as disturbances of memory and learning, schizophrenia, sexual disturbances, ischemic attacks, ictus, etc. For example, a compound according to formula (I): is administered to treat or prevent diseases of the central nervous system having a positive or negative modulation of AMPA/Kainate receptors and a negative modulation of NMDA receptors.
机译:2-氨基苯磺酰胺衍生物用于治疗或预防与谷氨酸能神经传递的正向或负向调节有关的中枢神经系统障碍,例如记忆和学习障碍,精神分裂症,性障碍,缺血性发作,黄疸等。例如,根据式(I)的化合物被施用以治疗或预防具有AMPA / Kainate受体的正或负调节和NMDA受体的负调节的中枢神经系统疾病。

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