首页> 外国专利> METHOD FOR TREATMENT AND PREVENTION OF DISTURBANCES OF THE CENTRAL NERVOUS SYSTEM ASSOCIATED WITH AN ALTERATION OF GLUTAMATERGIC NEUROTRANSMISSION BY ADMINISTRATION OF 2-AMINOBENZENESULFONAMIDE DERIVATIVES

METHOD FOR TREATMENT AND PREVENTION OF DISTURBANCES OF THE CENTRAL NERVOUS SYSTEM ASSOCIATED WITH AN ALTERATION OF GLUTAMATERGIC NEUROTRANSMISSION BY ADMINISTRATION OF 2-AMINOBENZENESULFONAMIDE DERIVATIVES

机译:通过管理2-氨基苯甲磺酰胺衍生物改变和调节谷氨酸神经发射而引起的中枢神经系统疾病的治疗和预防方法

摘要

2-aminobenzenesulfonamide derivatives are used to treat or prevent the interference of central nervous system, with positively or negatively adjusting Glutamatergic neurotransmission, such as memory disorders and association, schizophrenia, sexual harassment, ischemic challenge, breaking-out etc.. For example, compound is according to formula (I): giving and treat or prevent central nervous system with the negatively-modulated nmda receptor in positive or negative modulation AMPA/Kainate receptors.
机译:2-氨基苯磺酰胺衍生物用于治疗或预防中枢神经系统的干扰,通过正向或负向调节谷氨酸能神经传递,例如记忆障碍和联想,精神分裂症,性骚扰,缺血性发作,爆发等。例如,化合物根据式(I):用正或负调节的AMPA / Kainate受体中的负调节的nmda受体给予和治疗或预防中枢神经系统。

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