首页> 外国专利> PYRAZOLOPYRIDINE-4-YL PYRIDAZINONE DERIVATIVE AND ADDITION SALT THEREOF, AND PDE INHIBITOR COMPRISING THE DERIVATIVE OR SALT AS ACTIVE INGREDIENT

PYRAZOLOPYRIDINE-4-YL PYRIDAZINONE DERIVATIVE AND ADDITION SALT THEREOF, AND PDE INHIBITOR COMPRISING THE DERIVATIVE OR SALT AS ACTIVE INGREDIENT

机译:吡唑并吡啶-4-基吡嗪酮衍生物及其盐分,以及含有该衍生物或盐分作为活性成分的PDE抑制剂

摘要

[PROBLEMS] To provide a novel pyrazolopyridine-4-yl pyridazinone derivative which has a phosphodiesterase inhibitory activity and is useful as a therapeutic agent. [MEANS FOR SOLVING PROBLEMS] A pyrazolopyridine-4-yl pyridazinone derivative represented by the general formula (1) (e.g., 6-(2-ethyl-7-methoxy-pyarzolo[1,5-a]pyridine-4-yl)-5-methyl-4,5-dihydro-3(2H)-pyridazinone).
机译:[问题]提供一种新型的吡唑并吡啶-4-基哒嗪酮衍生物,其具有磷酸二酯酶抑制活性并且可用作治疗剂。 [解决问题的方法]由通式(1)表示的吡唑并吡啶-4-基哒嗪酮衍生物(例如6-(2-乙基-7-甲氧基-吡唑并[1,5-a]吡啶-4-基) -5-甲基-4,5-二氢-3(2H)-哒嗪酮)。

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