首页> 外国专利> USE OF 3-(1H-IMIDAZOL-4-YLMETHYL)-INDAN-5-OL IN THE MANUFACTURE OF A MEDICAMENT FOR INTRASPINAL, INTRATHECAL OR EPIDURAL ADMINISTRATION

USE OF 3-(1H-IMIDAZOL-4-YLMETHYL)-INDAN-5-OL IN THE MANUFACTURE OF A MEDICAMENT FOR INTRASPINAL, INTRATHECAL OR EPIDURAL ADMINISTRATION

机译:3-(1H-咪唑-4-甲基)-茚满-5-OL在制备用于脊髓内,鞘内或硬膜外给药的药物中的用途

摘要

The present invention relates to a method for obtaining analgesia by administering 3-(1H-imidazol-4-ylmethyl)-indan-5-ol, its enetiomer or pharmaceutically acceptable ester or salt thereof to a mammal intraspinally. 3-(1H-imidazol-4-ylmethyl)-indan-5-ol, its enantiomer or a pharmaceutically acceptable ester or salt thereof can be administered intraspinally to a mammal obtaining analgesia without side-effects, such as sedation. The present invention also relates to a method for using the drug as an adjunct to anaesthesia by administering it intraspinally.
机译:本发明涉及通过将3-(1H-咪唑-4-基甲基)-茚满-5-醇,其对映异构体或其药学上可接受的酯或盐给予哺乳动物脊髓内镇痛的方法。可以将3-(1H-咪唑-4-基甲基)-茚满-5-醇,其对映异构体或其药学上可接受的酯或盐脊髓内给药至获得镇痛作用的哺乳动物,而没有副作用例如镇静作用。本发明还涉及通过脊髓内给药将该药物用作麻醉的辅助方法。

著录项

  • 公开/公告号IL141680B

    专利类型

  • 公开/公告日2007-06-17

    原文格式PDF

  • 申请/专利权人 ORION CORPORATION;

    申请/专利号IL141680

  • 发明设计人

    申请日2001-02-27

  • 分类号C07D233/64;A61K31/4164;A61K31/4174;A61P23/00;A61P25/04;A61P25/28;

  • 国家 IL

  • 入库时间 2022-08-21 20:58:42

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