NON-IMIDAZOL ARYLOXIPIPERIDINE AS LEGANDS OF THE H3 RECEIVER.

摘要

A compound of ** formula **, where X is O; n is an integer from 0 to 3; R5 is C1-C10 alkyl, C3-C8 alkenyl, C3-C8 cycloalkyl, C3-C8 cycloalkyl C1-C6 alkyl, C1-C6 phenylalkyl, C3-C8 phenylalkyl, or C1-C8 alkylcarbonyl C1-C8 alkyl; one of R1, R2 and R3 is G or W, where one of the remaining two is selected from H and halogen and the third being hydrogen; G is one of the following nitrogen-containing groups: -OL1Q, -L2Q, -N (L1Q) R5, -L3C (L1Q) R6R7, -C (L1Q) R6R7; or a pharmaceutically acceptable salt, ester, or amide thereof.