首页> 外国专利> COMPOSITION COMPRISING 2',4',5,7-TETRAHYDROXY-5',6-DIPRENYL FLAVANONE COMPOUND SHOWING POTENT INHIBITING ACTIVITY OF TUMOR CELL PROPAGATION FOR THE PREVENTION AND TREATMENT OF CANCER DISEASE

COMPOSITION COMPRISING 2',4',5,7-TETRAHYDROXY-5',6-DIPRENYL FLAVANONE COMPOUND SHOWING POTENT INHIBITING ACTIVITY OF TUMOR CELL PROPAGATION FOR THE PREVENTION AND TREATMENT OF CANCER DISEASE

机译:包含2',4',5,7-四羟基-5',6-二甲苯基黄烷酮化合物的组合物显示出抑制肿瘤细胞增殖的活性,可预防和治疗癌症。

摘要

A pharmaceutical composition containing 2,4,5,7-tetrahydroxy-5,6-diprenyl flavanone compound extracted from root of Cudrania tricuspidata is provided to inhibit propagation of tumor cells due to kinase 2(CKII) inhibition effect, thereby being used as a pharmaceutical composition for preventing and treating cancer diseases. The pharmaceutical composition for preventing and treating cancer diseases comprises 2,4,5,7-tetrahydroxy-5,6-diprenyl flavanone compound having tumor cell propagation inhibiting activity and represented by the formula(1) or a pharmaceutically acceptable salt thereof as an effective ingredient.
机译:提供了一种药物组合物,该药物组合物包含从from木(Cudrania tricuspidata)的根中提取的2,4,5,7-四羟基-5,6-二异戊烯基黄烷酮化合物,以抑制由于激酶2(CKII)抑制作用而引起的肿瘤细胞的增殖,从而用作用于预防和治疗癌症疾病的药物组合物。预防和治疗癌症疾病的药物组合物包含有效的由式(1)表示的具有肿瘤细胞增殖抑制活性的2,4,5,7-四羟基-5,6-二异戊烯基黄烷酮化合物或其药学上可接受的盐。成分。

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