首页> 外国专利> TRANSDERMAL INTRODUCTION TO THE ORGANISM OF COMPLEX (R) -3, 3-DIPHENYLPROPYLAMINOMONOMETERS

TRANSDERMAL INTRODUCTION TO THE ORGANISM OF COMPLEX (R) -3, 3-DIPHENYLPROPYLAMINOMONOMETERS

机译:透皮法介绍复合物(R)-3,3-二苯丙胺基单体

摘要

The invention relates to a device for transdermally administering a compound of formula (I), wherein A represents hydrogen or deuterium, R represents a group selected among C1-4alkyl, C3-10cycloalkyl, or phenyl, each of which can be substituted by C1-3alkoxy, fluoride, chlorine, bromine, iodine, nitro, amino, hydroxy, oxo, mercapto, or deuterium, the C atom marked by * (asterisk) being provided in the R configuration. The invention is characterized in that the compound of general formula (I) is provided in a polymer matrix and is released at a dose of 0.5 to 20 mg per day through human skin. The invention further relates to the use of said compounds of formula (I) for producing transdermal medicaments.
机译:本发明涉及用于透皮给药式(I)化合物的装置,其中A代表氢或氘,R代表选自C1-4烷基,C3-10环烷基或苯基的基团,它们各自可以被C1-取代。 3烷氧基,氟化物,氯,溴,碘,硝基,氨基,羟基,氧代,巯基或氘代,以*(星号)标记的C原子以R构型提供。本发明的特征在于将通式(I)的化合物提供在聚合物基质中,并且每天以0.5至20mg的剂量通过人皮肤释放。本发明进一步涉及所述式(I)化合物在生产透皮药物中的用途。

著录项

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号