首页> 外国专利> Process for purifying N-3-(3-cyanopyrazolo1,5-apyrimidin-7-yl)phenyl-N-ethylacetamide(zaleplon) and crystalline forms of zaleplon accessible with the process

Process for purifying N-3-(3-cyanopyrazolo1,5-apyrimidin-7-yl)phenyl-N-ethylacetamide(zaleplon) and crystalline forms of zaleplon accessible with the process

机译:纯化N- [3-(3-氰基吡唑并[1,5-a]嘧啶-7-基)苯基] -N-乙基乙酰胺(扎来普隆)和扎来普隆的结晶形式的方法

摘要

Provided are novel Zaleplon crystalline Forms II, III, IV and V, which are useful for the treatment of insomnia. Also provided are processes for making Forms I, II, and V using precipitation methods.
机译:提供新颖的扎来普隆晶体形式II,III,IV和V,其可用于治疗失眠。还提供了使用沉淀法制备形式I,II和V的方法。

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