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Preparation, composition, and pharmaceutical use of new generation triple-sighted, chiral, broad spectrum antibacterial, 7-substituted piperidino-quinolone carboxylic acid derivatives

机译:新一代三目,手性,广谱抗菌,7位取代的哌啶子基-喹诺酮羧酸衍生物的制备,组成和药物用途

摘要

This invention relates to new generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, to their optical isomers, diastereomers or enantiomers, as well as pharmaceutically acceptable salts, hydrates, prodrugs, polymorphs and pseudopolymorphs thereof, to their preparation, to their compositions and to their use.
机译:本发明涉及新一代三靶向,手性,广谱抗微生物的7-取代哌啶子基-喹诺酮羧酸衍生物,涉及它们的旋光异构体,非对映异构体或对映异构体,及其药学上可接受的盐,水合物,前药,多晶型物和假多晶型物,其制备,组成和用途。

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