首页> 外国专利> ORTHO-SUBSTITUTED NITROGEN-CONTAINING BISARYL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS POTASSIUM CHANNEL INHIBITORS

ORTHO-SUBSTITUTED NITROGEN-CONTAINING BISARYL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS POTASSIUM CHANNEL INHIBITORS

机译:邻位取代的氮杂双芳基化合物,包含它们的药物组合物及其作为钾通道抑制剂的用途

摘要

Ortho, ortho-substituted nitrogen-containing bisaryl compounds, processes for their preparation, their use as medicaments, and pharmaceutical preparations including their use as antiarrhythmic active compounds, for example, for the treatment and prophylaxis of atrial arrhythmias, e.g. atrial fibrillation (AF) or atrial flutters. Compounds of the invention include compounds of the formula I
机译:邻位,邻位取代的含氮双芳基化合物,其制备方法,其用作药物的用途以及包括其作为抗心律不齐活性化合物的药物制剂的用途,例如,用于治疗和预防房性心律不齐,例如心房颤动(AF)或房扑。本发明的化合物包括式I的化合物

著录项

  • 公开/公告号IL156312B

    专利类型

  • 公开/公告日2009-05-04

    原文格式PDF

  • 申请/专利权人 SANOFI-AVENTIS DEUTSCHLAND GMBH;

    申请/专利号IL156312

  • 发明设计人

    申请日2003-06-04

  • 分类号C07D239/28;A61K31/4418;A61K31/444;A61K31/497;A61K31/505;A61K31/506;A61K45/00;A61P9/00;A61P9/06;A61P25/02;A61P43/00;C07D213/56;C07D213/81;C07D213/82;C07D241/24;C07D401/12;C07D401/14;C07D413/12;C07D413/14;

  • 国家 IL

  • 入库时间 2022-08-21 19:27:46

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