首页> 外国专利> Tiazoliloxifenilamidinas or tiadiazoliloxifenilamidinas and its use as Fungici - das

Tiazoliloxifenilamidinas or tiadiazoliloxifenilamidinas and its use as Fungici - das

机译:替硝唑西芬拉米达米纳斯或噻二唑西芬拉米达米纳斯及其作为真菌的用途-das

摘要

This also relates to a process for its preparation, the use of the amidines according this to combat unwanted Microorganisms, as well as an agent for this purpose, a procedure to combat unwanted microorganisms by application of the compounds according to the sun Icitud on microorganisms and / or their habitat.Claim 1: tiadiazoliloxifenilamidina or tiazoliloxifenilamidina of formula (1) which is and CR7 o n; n is an integer selected from 0, 1, 2, 3, 4 and 5; r1 is selected from Hydrogen, alkyl groups C1 - C2 - 12 12, alquenilo alquinilo C212, linear or branched, groups cyclic S for rent 12 alquenilo C3, C4 and C4 alquinilo - 12 12Where in the Ring System of all cyclic groups previously mentioned one or more C Atoms can be replaced with heteroatoms selected from N, o, P and S, and all groups previously mentioned may be substituted with one or More groups that are Selection By - R '- X, - -' Or '-' Sir 'nr 2, - 3, - coor - CN -, and conr2',Where R can be Hydrogen or an alkyl group C1 - 12, - SH, - sru00f6, where Ru00f6 alkyl group can be a linear or branched C1 - 12, which can be substituted with one or More groups that are selected - R '- X, - - or', 'Mr. id,' Sir '- 2, 3 - coor - CN -, and conr2', where r 'is the S Previous ignificados; R2 and R3 are independently selected from among themselves,The Group comprised 12 alkyl groups C1, C2 alquenilo alquinilo C2 - 12 - 12, linear or branched alkyl groups, cyclic alquenilo C4 C3 - 12, - 12, - 12 alquinilo C4, C5 aryl groups 18, 19 or alcarilo aralquilo C7 C7 - 19, where the Ring System all the cyclic groups previously Referred to one or more C Atoms can be replaced with heteroatoms selected from N, or,P and s groups and all the previously mentioned may be substituted with one or More groups that are selected - R '- X, - -' Or '-' Sir 'nr 2, - 3, - coor - CN -, and conr2', where r 'is the meanings above; or where the R2 and R3, R2 and R1 and R1 and R3 together with Atoms We are United with other Atoms or selected n, or,P and S can form a Ring of four to Seven members, which in turn can be substituted with one or More groups X, R ', or', '' Sir ', nr 2, 3, coor, cn and conr 2', where r 'is the old meanings; R4 and R5 are independently selected from the Group comprising it CN x, h, alkyl groups C1, C2 alquenilo - 12, - 12, - 12 alquinilo C2 linear or branchedCyclic alkyl groups alquenilo C4 C3 - 12, - 12, - 12 alquinilo C4, C5 aryl groups 18, 19 or alcarilo aralquilo C7 C7 - 19, where the Ring System of all cyclic groups previously mentioned one or more C Atoms can be replaced with heteroatoms selected from N, or,P and s groups and all the previously mentioned may be substituted with one or More groups that are selected - R '- X, - -' Or '-' Sir 'nr 2, - 3, - coor - CN -, and conr2', where r 'is the meanings previous; R6 is selected from the group consisting of - X, - CN, - SH, - sru00f6, - oru00f6, - (c = o) - Ru00f6 alkyl groups C1, C2 alquenilo - 12, - 12, - 12 alquinilo C2 linear or branchedCyclic alkyl groups alquenilo C4 C3 - 12, - 12, - 12 alquinilo C4, C5 aryl groups 18, 19 or alcarilo aralquilo C7 C7 - 19, where the Ring System of all cyclic groups previously mentioned one or more C Atoms can be replaced with heteroatoms selected from N, or,P and s groups and all the previously mentioned may be substituted with one or More groups that are selected - R '- X, - -' Or '-' Sir 'nr 2, - 3, - coor - CN -, and conr2', where r 'and Ru00f6 have previous meanings; and R7 is selected from the group consisting of - X, - CN, - SH Sru00f6 oru00f6, -, -, - (c = o) - Ru00f6 alkyl groups C1, C2 alquenilo - 12, - 12, - 12 alquinilo C2 linear or branchedCyclic alkyl groups alquenilo C4 C3 - 12, - 12, - 12 alquinilo C4, C5 aryl groups 18, 19 or alcarilo aralquilo C7 C7 - 19, where the Ring System of all cyclic groups previously mentioned one or more C Atoms can be replaced with heteroatoms selected from N, or,P and s groups and all the previously mentioned may be substituted with one or More groups that are selected - R '- X, - -' Or '-' Sir 'nr 2, - 3, - coor - CN -, and conr2', where r 'and Ru00f6 have previous meanings. Claim 7: alcohol; or tiadiazolilo of formula (2) in the R6, and N have the meanings above.Claim 1: tiadiazolilo thiazolyl or Derivative of formula (3), in which z is a group output, selected from the group consisting trifltato mesilate, tosylate, halogens, or so2me and R6, and N have the meanings above. Claim 1: ether - or tiadiazolilaminofenu00edlico thiazolyl and formula (4) in the R4 and R6, and N have the meanings above.Claim 1: ether - or tiadiazolilaminofenu00edlico thiazolyl and formula (5) in the R4 and R6, and N have the meanings above.
机译:这也涉及其制备方法,根据本发明的idine在对抗有害微生物方面的用途,以及用于该目的的试剂,通过将根据本发明的阳光化合物施用在微生物上来防治有害微生物的方法和方法。权利要求1:式(1)的噻二唑和苯并噻吩并在它们的CR7上存在; n是选自0、1、2、3、4和5的整数; r1选自氢,烷基C1-C2-12 12,直链或支链烷基,直链或支链的环烷基S出租12 alquenilo C3,C4和C4直链烷基-12 12其中,在所有环基的环系中,前面提到的一个可以用选自N,o,P和S的杂原子取代一个或多个C原子,并且前面提到的所有基团都可以被一个或多个选择为-R'-X,--'或'-'Sir的基团取代“ nr 2-3-coor-CN-和conr2”,其中R可以是氢或烷基C1-12,-SH,-sr u00f6,其中R u00f6烷基可以是直链或支链C1-12,其可以被一个或多个选择的基团取代-R'-X,-或','Mr。 id,'爵士'-2,3-coor-CN-和conr2',其中r'是S先前的ignificados; R 2和R 3彼此独立地选择。该基团包括12个烷基C 1,C 2烷基萘醌C 2-12-12,直链或支链烷基,环状烷基C 4 C 3-12 -12-12烷基萘4,C 5芳基第18、19或alcarilo aralquilo C7 C7-19族,其中环系统以前所有指的一个或多个C原子可被选自N,或P和s组的杂原子取代,并且所有先前提及的被一个或多个选择的基团取代-R'-X,--'或'-'Sir'nr 2,-3,-coor-CN-和conr2',其中r'是上面的含义;或其中R2和R3,R2和R1和R1和R3连同我们与其他原子或所选n结合的原子,或者,P和S可以形成四至七个成员的环,而该环又可以被一个取代或更多组X,R'或','Sir',nr 2、3,coor,cn和conr 2',其中r'是旧含义; R4和R5独立地选自包含CNx,h,烷基C1,C2的烷基萘基C12,C12、12、12 Alquinilo C2直链或支链的环状烷基Alquenilo C4 C3-12、12、12 Alquinilo C4 ,C5芳基18、19或alcarilo aralquilo C7 C7-19,其中先前提及的所有环基的环系统可将一个或多个C原子替换为选自N,P,s和所有前述基团的杂原子可以用一个或多个选择的基团取代-R'-X,--'或'-'Sir'nr 2-3,-coor-CN-和conr2',其中r'是先前的含义; R 6选自-X,-CN,-SH,-sr u00f6,-或 u00f6,-(c = o)-R u00f6烷基C1,C2烷基-12,-12,- 12个Alquinilo C2直链或支链环状烷基alquenilo C4 C3-12-12-12 alquinilo C4,C5芳基18、19或alcarilo aralquilo C7 C7-19,其中所有环状基团的环系统先前都提到一个或多个C原子可以被选自N,P和s组的杂原子取代,所有前面提到的原子都可以被一个或多个选定的基团取代-R'-X,--'或'-'Sir'nr 2 -3,-coor-CN-和conr2',其中r'和R u00f6具有先前含义; R7选自-X,-CN,-SH Sr u00f6或 u00f6,-,-,-(c = o)-R u00f6烷基C1,C2烷基-12,-12, -12个alquinilo C2直链或支链环状烷基alquenilo C4 C3---12--12 alquinilo C4,C5芳基18、19或alcarilo aralquilo C7 C7-19,其中所有环状基团的环系统先前都提到一个或多个C原子可以被选自N,P或s基团的杂原子取代,并且所有前面提到的原子都可以被一个或多个选定的基团取代-R'-X,--'或'-'Sir'nr 2 ,-3,-coor-CN-和conr2',其中r'和R u00f6具有先前的含义。要求7:酒精;权利要求1:式(3)的噻二唑噻唑基或衍生物,其中z是基团输出,选自甲磺酸三氟甲磺酸酯,甲苯磺酸酯,卤素,或so2me和R6,以及N具有上述含义。权利要求1:R4和R6中的醚-或噻二唑胺基氨基噻吩并噻唑基和式(4),并且N具有上述含义。权利要求1:R4和R6的醚-或噻二唑胺基氨基苯甲酸噻唑基和式(5),以及N具有上述含义。

著录项

  • 公开/公告号AR069707A1

    专利类型

  • 公开/公告日2010-02-10

    原文格式PDF

  • 申请/专利权人 BAYER CROPSCIENCE AG;

    申请/专利号AR2008P105466

  • 发明设计人

    申请日2008-12-16

  • 分类号C07D277/34;C07D285/08;C07D417/12;A01N43/78;A01N43/836;

  • 国家 AR

  • 入库时间 2022-08-21 18:47:33

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