首页> 外国专利> 2- 4- (PYRAZOL-4-ILALKIL) PIPERAZIN-1-IL -3-PHENYL PIRASINES AND PYRIDINES AND 3- 4- (PYRAZOL-4-ILALKIL) PIPERAZIN-1-IL -2-PHENYL-Pyrynyl QUALITY OF ANTAGONISTS OF 5-HT RECEPTORS

2- 4- (PYRAZOL-4-ILALKIL) PIPERAZIN-1-IL -3-PHENYL PIRASINES AND PYRIDINES AND 3- 4- (PYRAZOL-4-ILALKIL) PIPERAZIN-1-IL -2-PHENYL-Pyrynyl QUALITY OF ANTAGONISTS OF 5-HT RECEPTORS

机译:2- [4-(吡唑-4-吡咯)哌嗪-1-IL] -3-苯基哌嗪和吡啶和3- [4-(吡唑-4-吡咯)哌嗪-1-IL] -2-苯基嘧啶5-HT受体拮抗剂的质量

摘要

The present invention provides compounds of formula I, which are selective 5-HT receptor antagonists, and their use in the treatment of migraine, persistent pain and anxiety, where each of A and B is independently —C (H) = or —N =, provided that at least one of A and B is —N =, n is 1-3, m is 0-3, and R are as defined herein.
机译:本发明提供了作为选择性5-HT受体拮抗剂的式I化合物,及其在治疗偏头痛,持续性疼痛和焦虑中的用途,其中A和B各自独立地为-C(H)=或-N =假设A和B中的至少一个是-N =,n是1-3,m是0-3,并且R如本文所定义。

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