首页> 外国专利> BICYCLIC COMPOUND AS SELECTIVE MELANIN-CONCENTRATING HORMONE RECEPTOR ANTAGONIST FOR TREATING OBESITY AND RELATED DISORDER

BICYCLIC COMPOUND AS SELECTIVE MELANIN-CONCENTRATING HORMONE RECEPTOR ANTAGONIST FOR TREATING OBESITY AND RELATED DISORDER

机译:双环化合物作为治疗肥胖症及相关疾病的选择性黑色素浓缩激素受体拮抗剂

摘要

PROBLEM TO BE SOLVED: To provide a method for preparing an antagonistic compound against a melanin-concentrating hormone, and to provide a method for using the compound in the treatments of metabolic disorders and eating disorders (e.g. obesity, diabetes).SOLUTION: The new bicyclic compound having MCH (melanin-concentrating hormone) antagonistic activity is provided, which is represented by formula 3.
机译:解决的问题:提供一种制备针对黑色素浓缩激素的拮抗化合物的方法,并提供将该化合物用于代谢性疾病和饮食失调(例如肥胖症,糖尿病)的治疗方法。提供了具有MCH(黑色素浓缩激素)拮抗活性的双环化合物,其由式3表示。

著录项

  • 公开/公告号JP2011006469A

    专利类型

  • 公开/公告日2011-01-13

    原文格式PDF

  • 申请/专利权人 PHARMACOPEIA DRUG DISCOVERY INC;

    申请/专利号JP20100200393

  • 发明设计人 GUO TAO;GU HUIZHONG;HOBBS DOUGLAS WALSH;

    申请日2010-09-07

  • 分类号C07D213/75;A61P43;A61P3;A61P3/04;A61P3/10;A61P25;A61K31/495;A61K31/496;C07D405/14;C07D401/12;C07D405/12;

  • 国家 JP

  • 入库时间 2022-08-21 18:25:17

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