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MOLECULAR MODULATORS OF THE WNT/BETA-CATENIN PATHWAY

机译:WNT /贝塔-连环蛋白通路的分子调节剂

摘要

The present invention is directed toward a method of treating a subject for a condition mediated by aberrant Wnt/β-catenin signaling by selecting a subject with a condition mediated by aberrant Wnt/β-catenin signaling and administering to the selected subject at least one compound selected from the group consisting of those set forth in Table 1, Table 2, Table 3, and a pharmaceutically acceptable salt thereof. A method of similarly modulating the Wnt/β-catenin pathway in a subject is also discussed.
机译:本发明涉及一种通过选择具有由Wnt /β-连环蛋白信号转导介导的病症的对象并向所选对象施用至少一种化合物来治疗由Wnt /β-连环蛋白信号转导介导的病症的对象的方法。选自表1,表2,表3中所列的那些及其药学上可接受的盐。还讨论了类似地调节受试者中的Wnt /β-连环蛋白途径的方法。

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