首页> 外国专利> MOLECULAR ACTIVATORS OF THE WNT/BETA-CATENIN PATHWAY

MOLECULAR ACTIVATORS OF THE WNT/BETA-CATENIN PATHWAY

机译:WNT /贝塔-连环蛋白通路的分子激活剂

摘要

The present invention is directed toward a method of treating a subject for a condition mediated by aberrant Wnt/β-catenin signaling by selecting a subject with a condition mediated by aberrant Wnt/β-catenin signaling and administering to the selected subject a compound selected from the group consisting of those set forth in Table 1, Table 2, and a pharmaceutically acceptable salt thereof. A method of similarly modulating the Wnt/β-catenin pathway in a subject is also discussed.
机译:本发明涉及一种通过选择具有由Wnt /β-连环蛋白信号转导介导的病症的对象并向所选对象施用选自以下的化合物来治疗由Wnt /β-连环蛋白信号转导介导的病症的对象的方法。表1,表2中列出的那些,及其药学上可接受的盐。还讨论了类似地调节受试者中的Wnt /β-连环蛋白途径的方法。

著录项

  • 公开/公告号US2017049793A1

    专利类型

  • 公开/公告日2017-02-23

    原文格式PDF

  • 申请/专利号US201514701936

  • 申请日2015-05-01

  • 分类号A61K31/708;A61K31/353;A61K31/7048;A61K31/357;A61K31/506;A61K31/4406;A61K31/167;A61K31/196;A61K31/24;A61K31/4409;A61K31/472;A61K31/5377;A61K31/69;A61K31/15;A61K31/495;A61K31/426;A61K31/52;A61K31/404;A61K31/405;A61K31/4178;A61K31/4439;A61K31/047;A61K31/695;A61K31/407;A61K31/403;A61K31/421;A61K31/5383;A61K31/351;A61K31/4152;A61K31/166;A61K31/585;A61K31/57;A61K31/565;A61K31/365;A61K31/201;A61K31/336;A61K31/4402;A61K31/015;A61K31/366;A61K31/553;A61K31/5575;A61K31/55;A61K31/27;A61K31/4245;A61K31/352;

  • 国家 US

  • 入库时间 2022-08-21 13:50:28

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