首页> 外国专利> NOVEL FUSED BRIDGED BICYCLIC HETEROARYL SUBSTITUTED 6-ALKYLIDENE PENEMS AS POTENT BETA-LACTAMASE INHIBITORS

NOVEL FUSED BRIDGED BICYCLIC HETEROARYL SUBSTITUTED 6-ALKYLIDENE PENEMS AS POTENT BETA-LACTAMASE INHIBITORS

机译:新型融合桥联双环杂芳基取代的6-亚烷基烯酮作为潜在的β-内酰胺酶抑制剂

摘要

A compound of formula (I) or formula (Ia); embedded image ;Wherein R1, Ra, R2, X, R3, Y1, Y2, A, B and C are as defined herein. Also, pharmaceutical compositions comprising such compounds and excipients, methods of treating bacterial infections comprising administering such compounds, methods for making such compounds and hydrates of such compounds.
机译:式(I)或式(Ia)的化合物; “嵌入式图像” ;其中R 1 ,R a ,R 2 ,X,R 3 ,Y 1 < / Sub>,Y 2 ,A,B和C如本文所定义。同样,包含此类化合物和赋形剂的药物组合物,治疗细菌感染的方法包括施用此类化合物,制备此类化合物的方法和此类化合物的水合物。

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