首页> 外国专利> NAPHTYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PHOSPHODIESTERASE ISOENZYME 4 (PDE4) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

NAPHTYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PHOSPHODIESTERASE ISOENZYME 4 (PDE4) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

机译:萘啶衍生物,其制备及其作为磷酸酯酶同工酶4(PDE4)抑制剂和含有它们的药物组合物的用途

摘要

The invention relates to compounds of formula I in free or salt form, where RSUP1 /SUPis a monovalent aromatic group having up to 10 carbon atoms, and RSUP2 /SUPis a cycloaliphatic group having up to 8 ring carbon atoms. Compositions containing them, methods for their preparation and their use as pharmaceuticals are also described.
机译:本发明涉及游离形式或盐形式的式I化合物,其中R 1 是具有至多10个碳原子的单价芳族基团,R 2 是脂环族基团具有最多8个环碳原子。还描述了包含它们的组合物,其制备方法及其在药物中的用途。

著录项

  • 公开/公告号HU0402311A3

    专利类型

  • 公开/公告日2012-03-28

    原文格式PDF

  • 申请/专利权人 NOVARTIS AG.;

    申请/专利号HU20040002311

  • 发明设计人

    申请日2002-11-04

  • 分类号A61K31/4375;A61P1/04;A61P1/12;A61P1/16;A61P3/10;A61P3/14;A61P7;A61P7/06;A61P9/04;A61P9/10;A61P9/12;A61P11;A61P11/04;A61P17;A61P17/12;A61P19/08;A61P19/10;A61P21/02;A61P21/04;A61P25;A61P25/16;A61P25/24;A61P25/28;A61P27/02;A61P27/16;A61P29;A61P35;A61P37;A61P37/02;A61P37/06;A61P37/08;A61P43;C07D471/04;

  • 国家 HU

  • 入库时间 2022-08-21 17:24:54

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