首页> 外国专利> DERIVATIVES OF 6-CYCLOAMINO-2-THIENYL-3-(PYRIDIN-4-YL)IMIDAZO1,2-B-PYRIDAZINE AND 6-CYCLOAMINO-2-FURANYL-3-(PYRIDIN-4-YL)IMIDAZO1,2-B-PYRIDAZINE, PREPARATION AND THERAPEUTIC APPLICATION THEREOF

DERIVATIVES OF 6-CYCLOAMINO-2-THIENYL-3-(PYRIDIN-4-YL)IMIDAZO1,2-B-PYRIDAZINE AND 6-CYCLOAMINO-2-FURANYL-3-(PYRIDIN-4-YL)IMIDAZO1,2-B-PYRIDAZINE, PREPARATION AND THERAPEUTIC APPLICATION THEREOF

机译:6-环氨基-2-噻吩-3-(吡啶-4-基)咪唑[1,2-B]-吡嗪和6-环氨基-2-呋喃基-3-(吡啶-4-基)咪唑的衍生物[1] ,2-B]-哒嗪,制备及其治疗应用

摘要

The invention relates to derivatives of 6-cycloamino-2-thienyl-3-(pyridin-4-yl)imidazo[1,2-b]-pyridazine and 6-cycloamino -2-furanyl-3-(pyridin-4-yl)imidazo[1,2-b]-pyridazine with general formula (I). The invention also relates to a method for the preparation and therapeutic application thereof, in the treatment or prevention of illnesses involving casein kinase 1 epsilon and/or casein kinase 1 delta.
机译:本发明涉及6-环氨基-2-噻吩-3-(吡啶-4-基)咪唑并[1,2-b]-哒嗪和6-环氨基-2-呋喃基-3-(吡啶-4-基)的衍生物通式(I)的咪唑并[1,2-b]-哒嗪。本发明还涉及用于制备或治疗应用的方法,其用于治疗或预防涉及酪蛋白激酶1ε和/或酪蛋白激酶1δ的疾病。

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