首页> 外国专利> PHARMACEUTICALLY ACCEPTABLE SALTS OF METHYL (3-{ 3-(6- AMINO- 2-BUTOXY-8-OXO-7, 8-DIHYDRO-9H-PURIN-9-YL) PROPYL (3- MORPHOLIN-4-YLPROPYL) AMINO METHYL } PHENYL) ACETATE AND THEIR USE IN THERAPY

PHARMACEUTICALLY ACCEPTABLE SALTS OF METHYL (3-{ 3-(6- AMINO- 2-BUTOXY-8-OXO-7, 8-DIHYDRO-9H-PURIN-9-YL) PROPYL (3- MORPHOLIN-4-YLPROPYL) AMINO METHYL } PHENYL) ACETATE AND THEIR USE IN THERAPY

机译:甲基(3- {[[[3-(6-氨基2-BUTOXY-8-OXO-7,8-DIHYDRO-9H-PURIN-9-YL)丙基](3-吗啉-4-基丙基)的药物可接受的盐)氨基}甲基}苯基)乙酸酯及其在治疗中的用途

摘要

Disclosed is a hydrochloric acid, hydrobromic acid or maleic acid salt of methyl (3- { [[3-(6-amino-2-butoxy-8-oxo-7, 8-dihydro-9H-purin-9-yl)propyl] (3-morpholin-4-ylpropyl)amino]- methyl} phenyl)acetate or a solvate of the salt for the treatment of asthma, COPD, allergic rhinitis, allergic conjunctivitis, atopic dermatitis, cancer, hepatitis B, hepatitis C, HIV, HPV, bacterial infections or dermatosis.
机译:公开了甲基(3-{[[[3-(6-氨基-2-丁氧基-8-氧代-7,8-二氢-9H-嘌呤-9-基)丙基]的盐酸,氢溴酸或马来酸盐。 ](3-吗啉-4-基丙基)氨基]-甲基}苯基)乙酸盐或盐的溶剂化物,用于治疗哮喘,COPD,过敏性鼻炎,过敏性结膜炎,特应性皮炎,癌症,乙型肝炎,丙型肝炎,HIV ,HPV,细菌感染或皮肤病。

著录项

  • 公开/公告号NZ585961A

    专利类型

  • 公开/公告日2012-05-25

    原文格式PDF

  • 申请/专利号NZ20080585961

  • 发明设计人 MCINALLY THOMAS;SCHULZ HAKAN;

    申请日2008-12-16

  • 分类号C07D473/18;A61K31/5377;A61P11;A61P11/06;A61P17;A61P31/12;A61P31/18;A61P35;A61P37/02;A61P37/08;

  • 国家 NZ

  • 入库时间 2022-08-21 17:23:26

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