首页> 外国专利> NEW BENZATHINE SALTS OF ACE INHIBITORS, PROCESS FOR THEIR PREPARATION AND THEIR USE FOR THE TREATMENT OF CARDIOVASCULAR DISEASES

NEW BENZATHINE SALTS OF ACE INHIBITORS, PROCESS FOR THEIR PREPARATION AND THEIR USE FOR THE TREATMENT OF CARDIOVASCULAR DISEASES

机译:ACE抑制剂的新苄沙丁胺盐,其制备方法及其在治疗心血管疾病中的用途

摘要

The present invention describes new salts of ACE inhibitors with N,N-dibenzylethylenediamine (abbr.: benzathine salts), a process for their preparation in crystal and amorphous forms by the reaction of two moles of ACE inhibitors with one mole of N,N-dibenzylethylenediamine, a process for the preparation of pharmaceutical formulations containing these salts and their use for the treatment of cardiovascular diseases.
机译:本发明描述了ACE抑制剂与N,N-二苄基乙二胺的新盐(缩写:苄星盐),其通过使两摩尔ACE抑制剂与一摩尔N,N-反应而制备成晶体和无定形形式的方法。二苄基乙二胺,一种含有这些盐的药物制剂的制备方法及其在治疗心血管疾病中的用途。

著录项

  • 公开/公告号IN2012CN03490A

    专利类型

  • 公开/公告日2013-07-26

    原文格式PDF

  • 申请/专利权人

    申请/专利号IN3490/CHENP/2012

  • 发明设计人 RUCHMAN RUDOLF;ZUPET PAVEL;

    申请日2012-04-18

  • 分类号C07D209/42;A61K31;A61P9/10;A61K31/551;C07D207/16;A61P9;A61K31/675;C07D209/52;A61K45/06;C07D209;C07D487/04;A61P9/12;A61K31/401;A61K31/403;

  • 国家 IN

  • 入库时间 2022-08-21 16:41:06

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