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NEW CHIRAL INTERMEDIATE, METHOD OF PRODUCING THEREOF AND ITS USE IN THE MANUFACTURE OF TOLTERODINE, FESOTERODINE, OR THE ACTIVE METABOLITE THEREOF
NEW CHIRAL INTERMEDIATE, METHOD OF PRODUCING THEREOF AND ITS USE IN THE MANUFACTURE OF TOLTERODINE, FESOTERODINE, OR THE ACTIVE METABOLITE THEREOF
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机译:新的手性中间体,其制备方法及其在制备托特罗定,非索达定或活性代谢物中的用途
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摘要
The compound of formula (I): is provided. It may be produced by subjecting a compound of formula (IV) to a reduction reaction wherein R represents hydrogen, straight or branched C1-C6 alkyl. This compound is a valuable intermediate which may be used in the synthesis of fesoterodine, tolterodine, its active metabolite, and related compounds.
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