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Compound having detrusor muscle-contracting activity and urethral sphincter muscle-relaxing activity
Compound having detrusor muscle-contracting activity and urethral sphincter muscle-relaxing activity
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机译:具有逼尿肌收缩活性和尿道括约肌松弛活性的化合物
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摘要
Disclosed is a compound represented by general formula (I) (wherein all of the symbols are as defined in the description), a salt or solvate of the compound, or a prodrug of the compound or the salt or solvate, a mixture of the compound with a diastereomer thereof at an arbitral ratio, or a cyclodextrin inclusion compound of the compound, which has a detrusor muscle-contracting activity and a urethral sphincter muscle-relaxing activity, and therefore can ameliorate bladder contraction disorders and/or urethral relaxation disorders, and is effective on, for example, underactive bladder. The compound has no risk of adverse side effects on a urinary system, a circulatory system and a digestive system, and has excellent pharmacokinetics including oral absorbability. As mentioned above, the compound is useful as a superior prophylactic, therapeutic and/or condition-ameliorating agent for underactive bladder.
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