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PEPTIDE, POLYNUCLEOTIDE, VECTOR, TRANSFORMANT, NFκB INHIBITOR, AND THERAPEUTIC AGENT FOR DISEASES ASSOCIATED WITH ACCELERATED NFκB ACTIVITY
PEPTIDE, POLYNUCLEOTIDE, VECTOR, TRANSFORMANT, NFκB INHIBITOR, AND THERAPEUTIC AGENT FOR DISEASES ASSOCIATED WITH ACCELERATED NFκB ACTIVITY
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机译:促进NFκB活性相关的疾病的肽,多核苷酸,矢量,转化子,NFκB抑制剂和治疗剂
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摘要
This peptide has an NFκB inhibitory effect and is any one of the following peptides: (a) a peptide comprising any amino acid sequence from SEQ ID NOs: 1-5; (b) a peptide having an NFκB inhibitory effect and comprising any amino acid sequence from SEQ ID NOs: 1-5, wherein one or a plurality of amino acid residues having been replaced, deleted and/or added; (c) a peptide having an NFκB inhibitory effect and comprising an amino acid sequence that is at least 80% homologous with any amino acid sequence from SEQ ID NOs: 1-5; (d) a peptide in which a cell-penetrating peptide is fused with any peptide selected from (a)-(c); and (e) a peptide in which a Met residue, a MetAla residue or an Ala residue is added to the N terminal of any peptide selected from (a)-(d).
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机译:该肽具有NFκB抑制作用,并且是以下肽中的任何一种:(a)包含来自SEQ ID NO:1-5的任何氨基酸序列的肽; (b)具有NFκB抑制作用的肽,其包含SEQ ID NO:1-5的任何氨基酸序列,其中一个或多个氨基酸残基已被替换,缺失和/或添加; (c)具有NFκB抑制作用的肽,其包含与SEQ ID NO:1-5的任何氨基酸序列至少80%同源的氨基酸序列; (d)一种肽,其中将穿透细胞的肽与选自(a)-(c)的任何肽融合; (e)一种肽,其中Met残基,MetAla残基或Ala残基被添加至选自(a)-(d)的任何肽的N末端。
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