首页> 外国专利> CENTRAL NERVOUS SYSTEM CELL PROTECTANT, AND AGENT FOR PREVENTION OR TREATMENT OF CENTRAL NERVOUS SYSTEM DEGENERATIVE DISEASE

CENTRAL NERVOUS SYSTEM CELL PROTECTANT, AND AGENT FOR PREVENTION OR TREATMENT OF CENTRAL NERVOUS SYSTEM DEGENERATIVE DISEASE

机译:中枢神经系统细胞保护剂,以及预防或治疗中枢神经系统退行性疾病的治疗剂

摘要

PROBLEM TO BE SOLVED: To provide a novel central nervous system cell protectant comprising galacto-N-biose, lacto-N-biose I, or their derivatives as an active ingredient, and an agent for the prevention or treatment of central nervous system degenerative disease.;SOLUTION: The present invention provides a compound represented by formula (1) or (2) or a pharmacologically acceptable salt thereof, or their prodrugs (R1s independently represent a halogen atom, an alkyl group, an alkenyl group, an aryl group, a cyano group, -N(R2)2, -NHCOR3, or -OR4; R2s independently represent H or an alkyl group).;SELECTED DRAWING: Figure 2;COPYRIGHT: (C)2017,JPO&INPIT
机译:解决的问题:提供一种新颖的中枢神经系统细胞保护剂,其包含半乳糖-N-二糖,乳酸-N-二糖I或其衍生物作为有效成分,以及用于预防或治疗中枢神经系统退行性疾病的药剂。解决方案:本发明提供了由式(1)或(2)表示的化合物或其药理学上可接受的盐,或其前药(R 1 独立地表示卤原子,烷基,烯基,芳基,氰基,-N(R 2 2 ,-NHCOR 3 或-OR < Sup> 4 ; R 2 s独立代表H或烷基).;部分附图:图2;版权:(C)2017,JPO&INPIT

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