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Piridoncarboxamidas selected or its Salts as active substances of Plants Against abiotic stress

机译:选择Piridoncarboxamidas或其盐作为植物抗非生物胁迫的活性物质

摘要

These compounds are used to increase the Tolerance against abiotic stress in Plants to enhance Plant Growth and / or to increase the yield of plants.Claim 1: the use of piridincarboxamidas replaced the General formula (1) or salts thereof, for Increasing the Tolerance against abiotic stress in plants, where cu2083u208bu2086 - ru00b9 represents cycloalkyl, aryl or hetarilo, where each of these three radical is not replaced O radical is substituted with one or more selected from Halogen, Nitro, cyano, Hydroxy, nru2078ru2079,Cu2081u208bu2084 alkyl, alkoxy cu2081u208bu2084 haloalquilo cu2081u208bu2084 -, -, - haloalcoxi cu2081u208bu2084, cu2081u208bu2084 - Alquiltio, cu2081u208bu2084 - alquilsulfoxi, cu2081u208bu2084 - alquilsulfona, cu2081u208bu2084 - haloalquiltio, cu2081u208bu2084 - haloalquilsulfoxi, cu2081u208bu2084 - haloalquilsulfona, cu2081u208bu2084 - alkoxy carbonyl, cu2081u208bu2084 - haloalcoxi ca Rbonilo, cu2081u208bu2084 - alquilcarboxi, cu2083u208bu2086 - cu2083u208bu2086 - cu2081u208bu2086 cycloalkyl alkyl, cycloalkyl, cu2081u208bu2084 - - - cu2081u208bu2084 carbonyl alkoxy alkyl, alkyl - hidroxicarbonilo, hidroxicarbonil cu2081u208bu2084,Ru2078ru2079n carbonyl; Ru00b2 represents Hydrogen; and ru00b3 and ru2074 independently represent Hydrogen, alkyl cu2081u208bu2081u2086, cu2082u208bu2081u2086 - alquenilo or cu2082u208bu2081u2086 - alquinilo, where each of the last 3 waste is not replaced or substituted with one or more radical s Selected from Halogen, Hydroxy, alkoxy cu2081u208bu2084 -, cyano -, cu2081u208bu2084 haloalcoxi, cu2081u208bu2084 Alquiltio cu2081u208bu2084 alquilamino -, -, -] - [cu2081u208bu2084 di alkyl aminoHidroxicarbonilo cu2081u208bu2084 alkoxy -, [] - [] - haloalcoxi cu2081u208bu2084 carbonyl, carbonyl, cu2083u208bu2086 - that is not substituted cycloalkyl, aryl, or is replaced, which is not replaced or substituted heteroaryl, or is replaced or not replaced heterociclilo, which is not Sustituid Or is replaced, or represent [cu2081u208bu2084 - alkoxy carbonyl carbonyl] -, [cu2081u208bu2084 alkoxy carbonyl] - - - - - cu2081u208bu2088 alkyl carbonylCu2081u208bu2081u2086 - alquilcarbonilo, cu2081u208bu2081u2086 - haloalquilcarbonilo represent cu2083u208bu2086 -, or cycloalkyl, cu2084u208bu2086 - cicloalquenilo, cu2083u208bu2086 - condensate cycloalkyl, who is in a position of the Ring with a ring carbocu00edclico saturated or unsaturated between 4 and 6 members, or cu2084u208bu2086 Cycle Alquenilo condensate, which is in a position of the Ring with a ring carbocu00edclico saturated or unsaturated between 4 and 6 membersWhere each of the last 4 waste is not replaced or residue is replaced with one or more selected from Halogen, Hydroxy alkyl, cyano, cu2081u208bu2084, cu2081u208bu2084 - haloalquilo, cu2081u208bu2084 - alkoxy -, cu2081u208bu2084 haloalcoxi, cu2081u208bu2084 - Alquiltio, cu2081u208bu2084 - alquilamino [cu2081u208bu2084 -, di Lquil] amino] -, [cu2081u208bu2084 - alkoxy carbonyl, carbonyl haloalcoxi cu2081u208bu2084 - [] - cu2083u208bu2086, cycloalkyl, aryl, which is not replaced or substitutedHeteroaryl, or is replaced or not replaced heterociclilo, that is not replaced or substituted aryl or heteroaryl, or represent, heterociclilo, where each of these three radical is not replaced or substituted with one or more radical selected from halu00f3gen Or, Nitro, cyano, nru2078ru2079, cu2081u208bu2084 Hydroxy alkyl, alkoxy cu2081u208bu2084 haloalquilo cu2081u208bu2084 -, -, - haloalcoxi cu2081u208bu2084,Cu2081u208bu2084 - Alquiltio, cu2081u208bu2084 - alquilsulfoxi, cu2081u208bu2084 - alquilsulfona, cu2081u208bu2084 - haloalquiltio, cu2081u208bu2084 - haloalquilsulfoxi, cu2081u208bu2084 - haloalquilsulfona, cu2081u208bu2084 - alkoxy carbonyl, carbonyl haloalcoxi cu2081u208bu2084 - - - - cu2083u208bu2086, cu2081u208bu2084 alquilcarboxi, cycloalkyl, cu2083u208bu2086 cycloalkyl - C u2081u208bu2086 alkyl, alkoxy carbonyl cu2081u208bu2084 cu2081u208bu2084 - - - - - cu2081u208bu2084 hidroxicarbonil hidroxicarbonilo alkyl, alkyl, ru2078ru2079n carbonyl, or ru00b3 represents Hydrogen,Cu2081u208bu2086 alkyl and ru2074 cu2081u208bu2086 represents alkyl, alkoxy cu2082u208bu2086 alqueniloxi cu2081u208bu2086 -, -, - or - cu2082u208bu2086 alquiniloxi cu2082u208bu2086 haloalcoxi or cu2081u208bu2086 - alkyl - or ru00b3 and ru2074 SOu2082, together with the N Atom that connects represent a natural amino acid residue at its Racemic form or in s US D and L forms of respectiveOr ru00b3 and ru2074 together with the N atom of the Heterocyclic Ring or a carbocu00edclico connects are between Four and eight members, in addition to the N Atom can contain additional heteroatoms in the ring, preferably up to two additional Ring heteroatoms selected from N, o and S, and is not replaced or substituted with one or more selected residues between HalogenCu2081u208bu2084 cu2081u208bu2084 - haloalquilo alkyl, alkoxy, cu2081u208bu2084 - [] - carbonyl, cu2081u208bu2084 - alkoxy -, cu2081u208bu2084 haloalcoxi, cu2081u208bu2084 Alquiltio hydroxy -, and a Heterocyclic Ring may contain an oxo Group N or ru00b3 and ru2074 together with the N Atom that connects represent the Group - n = cru2075 - nru2076 Ru2077, and where ru2075 represents Hydrogen or alkyl cu2081u208bu2086; ru2076 and ru2077 independently represent Hydrogen or - alkyl or cu2081u208bu2086, ru2076,Ru2077 form together with the N atom of the Heterocyclic Ring connects a preferably saturated with between five and seven members, such as piperidinilo, pirrolidinilo or morfolinilo; and ru2078 and ru2079 independently represent Hydrogen or - alkyl and N cu2081u208bu2086; representation NTA 0, 1 or 2.Claim 12: piridincarboxamidas replaced the formula (1) or salts thereof, where cu2083u208bu2086 - ru00b9 represents phenyl or cycloalkyl, hetarilo, where each of these three residues is not replaced or residue is replaced with one or more selected from Halogen, Nitro, Nru2078ru2079 Hydroxy alkyl, cyano, cu2081u208bu2084, cu2081u208bu2084 - haloalquilo, cu2081u208bu2084 - alkoxy -, cu2081u208bu2084 haloalcoxi, cu2081u208bu2084 - Alquiltio,Cu2081u208bu2084 - alquilsulfoxi, cu2081u208bu2084 - alquilsulfona, cu2081u208bu2084 - haloalquiltio, cu2081u208bu2084 - haloalquilsulfoxi, cu2081u208bu2084 - haloalquilsulfona, cu2081u208bu2084 - alkoxy carbonyl, carbonyl cu2081u208bu2084 - haloalcoxi, cu2081u208bu2084 - alquilcarboxi, cu2083u208bu2086 - cu2083u208bu2086 - cu2081u208bu2086 cycloalkyl alkyl, cycloalkyl, cu2081 u208bu2084 - - - cu2081u208bu2084 carbonyl alkoxy alkyl, alkyl - hidroxicarbonilo, hidroxicarbonil cu2081u208bu2084,Ru2078ru2079n carbonyl; Ru00b2 represents Hydrogen; and ru00b3 represents Ethyl; and ru2074 represents chu2082chu2082 - ru00b9u2070 and ru00b9u2070 cu2081u208bu2088 represents Hydrogen, alkyl, or cu2082u208bu2088 - alquenilo cu2082u208bu2088 - alquinilo, where each of the last 3 waste is not replaced or substituted with one or more S selected residues between Halogen, Hydroxy, alkoxy cu2081u208bu2084 -, cyano -, cu2081u208bu2084 haloalcoxi, cu2081u208bu2084 - Alquiltio, cu2081u208bu2084 - alquilamino,[] - cu2081u208bu2084 - amino alkyl, alkoxy hidroxicarbonilo, cu2081u208bu2084 - [] - [] - haloalcoxi cu2081u208bu2084 carbonyl, carbonyl, or represents cu2081u208bu2084 - [] - alkoxy carbonyl carbonyl, carbonyl alkoxy cu2081u208bu2084 [] - - - - cu2081u208bu2088 alkyl carbonyl, cu2081u208bu2081u2086 - alquilcarbonilo, cu2081u208bu2081u2086 - haloalquilcarbonilo or repres - IT cu2083u208bu2086 cycloalkyl,Cu2084u208bu2086 - cicloalquenilo where each of the last two mentioned waste is not replaced or residue is replaced with one or more selected from Halogen, Hydroxy alkyl, cyano, cu2081u208bu2084, cu2081u208bu2084 - haloalquilo, cu2081u208bu2084 - alkoxy -, cu2081u208bu2084 haloalcoxi, cu2081u208bu2084 - Alquiltio, Alquilamino cu2081u208bu2084 -, di - cu2081u208bu2084 [] - amino alkyl, alkoxy cu2081u208bu2084 - [] - [] - haloalcoxi cu2081u208bu2084 carbonyl, carbonyl, cu2083u208bu2086 cycloalkyl, phenyl -,Heterociclilo represents phenyl or heteroaryl heteroaryl, or, or heterociclilo, where each of these three radical is not replaced or substituted with one or more radical selected from Halogen, Nitro, cyano, nru2078ru2079, cu2081u208bu2084 Hydroxy alkyl, cu2081u208bu2084 - haloalquilo, cu2081u208b By Land. Cu2081u208bu2084 haloalcoxi alkoxy -, -, - Alquiltio cu2081u208bu2084, cu2081u208bu2084 - alquilsulfoxi, cu2081u208bu2084 - alquilsulfona, cu2081u208bu2084 - haloalquiltio,Cu2081u208bu2084 - haloalquilsulfoxi, cu2081u208bu2084 - haloalquilsulfona, cu2081u208bu2084 - alkoxy carbonyl, carbonyl cu2081u208bu2084 - haloalcoxi, cu2081u208bu2084 - alquilcarboxi, cu2083u208bu2086 - cu2083u208bu2086 - cu2081u208bu2086 cycloalkyl alkyl, cycloalkyl, cu2081u208bu2084 - - - cu2081u208bu2084 carbonyl alkoxy alkyl, - C hidroxicarbonilo, hidroxicarbonil u2081u208bu2084 alkyl and carbonyl, ru2078ru2079n; ru2078 and ru2079 independently represent Hydrogen or - alkyl cu2081u208bu2086.
机译:这些化合物用于提高植物对非生物胁迫的耐受性,从而增强植物的生长和/或提高植物的产量。权利要求1:使用派瑞丁羧酰胺替代了通式(1)或其盐,以提高耐受性对抗植物中的非生物胁迫,其中c u2083 u208b u20b-r u00b9代表环烷基,芳基或hetarilo,其中这三个自由基均未被取代,O自由基被选自卤素,硝基,氰基的一个或多个取代,羟基,nr u2078r u2079,C u2081 u208b u2084烷基,烷氧基c u2081 u208b u2084卤代alquilo c u2081 u208b u2084-,-,-卤代醇c u2081 u208b u2084,c u2081 u208b u2084-Alquiltio,c u2081 u208b u2084-alquilsulfoxi,c u2081 u208b u2084-alquilsulfona,c u2081 u208b u2084-haloalquiltio,c u2081 u208b u2084-haloalquilsulfoxi u208b u2084-卤代磺砜,c u2081 u208b u2084-羰基烷氧基,c u2081 u208b u2084-卤代alcoxi ca Rbonilo,c u2081 u208b u2084-alquilc arboxi,c u2083 u208b u2086-c u2083 u208b u2086-c u2081 u208b u2086环烷基烷基,环烷基,c u2081 u208b u2084---c u2081 u208b u2084羰基烷氧基烷基,烷基-hidroxicarbonilo,hidroxicarbonil c u2081 u208b u2084,R u2078r u2079n羰基; R u00b2代表氢;和r u00b3和r u2074分别代表氢,烷基c u2081 u208b u2081 u2086,c u2082 u208b u2081 u2086-alquenilo或c u2082 u208b u2081 u2086-alquinilo,其中每个最后3个废物没有被一个或多个自由基取代或取代。选自卤素,羟基,烷氧基c u2081 u208b u2084-,氰基-,c u2081 u208b u2084卤代醇,c u2081 u208b u2084 Alquiltio c u2081 u208b u2084 alquilamino-,-,-]-[c u2081 u208b u2084二烷基氨基Hidroxicarbonilo c u2081 u208b u2084烷氧基-,[]-[]-卤代alcoxi c u2081 u208b u2084羰基,羰基,未取代的环烷基,芳基或未取代的,未取代的或取代的杂芳基,或者已取代或未取代的杂环取代基或非必需的或代表[c u2081 u208b u2084-烷氧基羰基羰基]-,[c u2081 u208b u2084烷氧基羰基]-----c u2081 u208b u2088烷基羰基C u2081 u208b u2081 u2086- alquilcarbonilo,c u2081 u208b u 2081 u2086-卤代碳烯代表c u2083 u208b u2086-或环烷基,c u2084 u208b u2086-cicloalquenilo,c u2083 u208b u2086-缩合环烷基,在带有环的环位置在4至6个成员之间饱和或不饱和的carboc u00edclico,或在4至6个成员之间具有饱和或不饱和环状carboc u00edclico的环Alquenilo冷凝物,它位于环的位置4个废物未被替换或残渣被卤素,羟基烷基,氰基,c u2081 u208b u2084,c u2081 u208b u2084-卤代alquilo,c u2081 u208b u2084-烷氧基中的一种或多种选自,c u2081 u208b u2084晕厥,c u2081 u208b u2084-Alquiltio,c u2081 u208b u2084-alquilamino [c u2081 u208b u2084-,di Lquil]氨基]-,[c u2081 u208b u2084-烷氧基羰基,羰基卤代醇c u2081 u208b u2084-[]-c u2083 u208b u2086,未被取代或取代的杂芳基,或被取代或未被取代的环烷基取代的杂环基,即未被取代或取代的芳基或杂芳基,或代表杂环基,其中这三个基团均未被一个或多个选自以下的基团取代或取代:卤素,硝基,氰基,nr u2078r u2079 ,c u2081 u208b u2084羟基烷基,烷氧基c u2081 u208b u2084卤代alquilo c u2081 u208b u2084-,-,-卤代alcoxi c u2081 u208b u2084,C u2081 u208b u2084-Alquiltio ,c u2081 u208b u2084-alquilsulfoxi,c u2081 u208b u2084-alquilsulfona,c u2081 u208b u2084-haloalquiltio,c u2081 u208b u2084-haloalquilsulfoxi,c u2081 u2081 -u208lo al ,c u2081 u208b u2084-烷氧基羰基,羰基卤代醇c u2081 u208b u2084----c u2083 u208b u2086,c u2081 u208b u2084链烷烃,环烷基,c u2083 u208b u2086环烷基-C u2081 u208b u2086烷基,烷氧基羰基c u2081 u208b u2084 c u2081 u208b u2084-----c u2081 u208b u2084 hidroxicarbonil hidroxicarbonilo烷基,烷基,r u2078r u2079n羰基或r u00b3代表氢,C u2081 u208b u2086烷基,而r u2074 c u2081 u208b u2086代表烷基,烷氧基c u2082 u208b u2086烷氧基x , u2081 u208b u20b-,-,-或-c u2082 u208b u2086 alquiniloxi c u2082 u208b u2086卤代醇或c u2081 u208b u2086-烷基-或r u00b3和r u2074 SO u2082,以及连接的N原子代表天然氨基酸其外消旋形式的残基或各自的S D和L形式的Or或r与杂环基团的N原子或carbocedclico连接,除N原子外,在4至8个成员之间在环中可以包含其他杂原子,优选至多两个选自N,o和S的额外的环杂原子,并且不被卤素C u2081 u208b u2084 c u2081 u208b u2084-卤代铝烷基,烷氧基,c上的一个或多个选定残基取代或取代 u2081 u208b u2084-[]-羰基,c u2081 u208b u2084-烷氧基-,c u2081 u208b u2084卤代烷氧基,c u2081 u208b u2084羟基芳基和杂环可包含一个氧代基团N或r u00b3和r u2074以及连接的N Atom代表基团-n = cr u2075-nr u2076 R u2077,其中r u2075代表氢或烷基c u2081 u208b u2086; r u2076和r u2077独立地表示氢或-烷基或c u2081 u208b u2086,r u2076,R u2077形式与杂环的N原子一起连接,饱和原子优选为5至7个,如哌啶子诺,吡咯烷迪诺或吗啉代; r u2078和r u2079独立地表示氢或-烷基和N c u2081 u208b u2086;代表NTA 0、1或2。声明12:用piirdincarboxamidas取代了式(1)或其盐,其中c u2083 u208b u2086-r u00b9代表苯基或环烷基,杂多,其中这三个残基均未被取代或残基被一种或多种选自卤素,硝基,Nr u2078r u2079的羟基烷基,氰基,c u2081 u208b u2084,c u2081 u208b u2084-卤代基洛基,c u2081 u208b u2084-烷氧基-,c u2081 u208b u2084卤代alcoxi,c u2081 u208b u2084-Alquiltio,C u2081 u208b u2084-alquilsulfoxi,c u2081 u208b u2084-alquilsulfona,c u2081 u208b u2084 haloalquiltio,c u2081 u208b u2084-haloalquilsulfoxi,c u2081 u208b u2084-haloalquilsulfona,c u2081 u208b u2084-烷氧基羰基,羰基c u2081 u208b u2084-haloalcoxi,c u2081 u208b u2084 u2084-alquilcarboxi,c u2083 u208b u2086-c u2083 u208b u2086-c u2081 u208b u2086环烷基,环烷基,c u2081 u208b u2084---c u2081 u208b u2084羰基烷氧基烷基,烷基-Hidroxicarbonilo,Hidrox icarbonil c u2081 u208b u2084,R u2078r u2079n羰基; R u00b2代表氢; r u00b3代表乙基;并且r u2074代表ch u2082ch u2082-r u00b9 u2070,而r u00b9 u2070 c u2081 u208b u2088代表氢,烷基或c u2082 u208b u2088-阿奎尼洛c u2082 u208b u2088-alquinilo,其中最后3个废物中的每一个都不被卤素,羟基,烷氧基c u2081 u208b u2084-,氰基-,c u2081 u208b u2084卤代醇, c u2081 u208b u2084-Alquiltio,c u2081 u208b u2084-alquilamino,[]-c u2081 u208b u2084-氨基烷基,烷氧基羟基碳酸氢盐,c u2081 u208b u2084-[]-[] -卤代醇c u2081 u208b u2084羰基,或代表c u2081 u208b u2084-[]-烷氧基羰基羰基,羰基烷氧基c u2081 u208b u2084 []-----c u2081 u208b u2088烷基羰基,c u2081 u208b u2081 u2086-alquilcarbonilo,c u2081 u208b u2081 u2086-卤代alalcarbonilo或代表-IT c u2083 u208b u2086环烷基,C u2084 u208b u2086-cicloalquen最后提到的两个废物中的每一个都没有被替换或残留物是替换为卤素,羟基烷基,氰基,c u2081 u208b u2084,c u2081 u208b u2084-卤代alquilo,c u2081 u208b u2084-烷氧基-,c u2081 u208b u2084中的一种或多种haloalcoxi,c u2081 u208b u2084-Alquiltio,Alquilamino c u2081 u208b u2084-,di-c u2081 u208b u2084 []-氨基烷基,烷氧基c u2081 u208b u2084-[]-[ ]-卤代烷氧基c u2081 u208b u2084羰基,羰基,c u2083 u208b u2086环烷基,苯基-,Herocicliclilo代表苯基或杂芳基杂芳基,或或,或杂环基,其中这三个基团中的每一个都不被取代或取代一个或多个选自卤素,硝基,氰基,nr 2078r 2097羟基烷基,c 20208 1208的卤代烷基,halalalquilo,陆地上的c2081208。 C u2081 u208b u2084卤代烷氧基烷氧基-,-,-Alquiltio c u2081 u208b u2084,c u2081 u208b u2084-Alquilsulfoxi,c u2081 u208b u2084-alquilsulfona,c u2081 u208b u208b -Halalalquiltio,C u2081 u208b u2084-Halalalquilsulfoxi,c u2081 u208b u2084-Halalalquilsulfona,c u2081 u208b u2084-烷氧基羰基,羰基c u2081 u208b u2084-haloalcoxi,c u2084-alquilcarboxi,c u2083 u208b u2086-c u2083 u208b u2086-c u2081 u208b u2086环烷基,环烷基,c u2081 u208b u2084---c u2081 u208b u2084羰基烷氧基烷基,-Chidroxicarbonilo,hidroxicarbil u2081 u208b u2084烷基和羰基,r u2078r u2079n; r u2078和r u2079独立地表示氢或烷基c u2081 u208b u2086。

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