首页> 外国专利> The high concentration of AP, keytika, at, CD20 and alpha include the alpha, tau, sigma, Omega, alpha, kappa, and alpha

The high concentration of AP, keytika, at, CD20 and alpha include the alpha, tau, sigma, Omega, alpha, kappa, and alpha

机译:AP,keytika,at,CD20和alpha的高浓度包括alpha,tau,sigma,Omega,alpha,kappa和alpha

摘要

The present invention relates to an antibody to the active [phi] alpha [phi] P [alpha] a [phi] a [phi] a [alpha] kappa] e [CD20] in a high concentration pharmaceutical preparation, for example. Rituximab, _kappa p p p p a lambda__mu_ pi_, or a mixture of Hu muab CD20 antibodies, or subcutaneous injection.In particular, the preparations of the invention include at least one effective dose of CD20 antibody. A preparation used as a combination of_alpha lambda_rho__delta__in an enzyme preparation to form one or more active substances. In addition, the preparation includes at least one regulatory factor, for example.A mixture of buffering factor X histidine, stabilizer, or stabilizer (e.g. two or more_alpha kappa_alpha rho_stabilizers). Trehalose dihydrate (a-a or sucrose and optional second methionine) as a nonionic surfactant, stabilizer, and an effective slope At least one enzyme is supplied.The preparation method and application of the preparation are provided.
机译:例如,本发明涉及针对高浓度药物制剂中的活性φαφPααφaακe [CD20]的抗体。利妥昔单抗,λ或Hu muab> CD20抗体的混合物,或皮下注射。特别地,本发明的制剂包括至少一种有效剂量的CD20抗体。一种在酶制剂中用作αλδ组合的制剂,可形成一种或多种活性物质。另外,所述制剂包括至少一种调节因子,例如,缓冲因子X组氨酸,稳定剂或稳定剂(例如两种或更多种α-κ-rho-稳定剂)的混合物。作为非离子表面活性剂,稳定剂和有效斜率的海藻糖二水合物(α-α或蔗糖和可选的第二甲硫氨酸),至少提供一种酶。提供了制备方法和该制剂的用途。

著录项

  • 公开/公告号CY1117941T1

    专利类型

  • 公开/公告日2017-05-17

    原文格式PDF

  • 申请/专利权人 F. HOFFMANN-LA ROCHE AG;

    申请/专利号CY201611000610T

  • 申请日2016-07-01

  • 分类号A61K9/19;A61K9;A61K38/47;A61K39;A61K39/395;A61K45/06;A61K47/10;A61K47/18;A61K47/20;A61K47/22;A61K47/26;C07K16/28;

  • 国家 CY

  • 入库时间 2022-08-21 13:39:37

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