首页> 外国专利> BENZIMIDAZOLE AND IMADAZOPYRIDINE CARBOXIMIDAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF INDOLEAMINE 2,3-DIOXYGENASE

BENZIMIDAZOLE AND IMADAZOPYRIDINE CARBOXIMIDAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF INDOLEAMINE 2,3-DIOXYGENASE

机译:苯并咪唑和咪唑并吡啶羧酰亚胺的化合物具有抑制吲哚并胺2,3-二氧合酶的活性

摘要

PROBLEM TO BE SOLVED: To provide indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors for treating cancer, viral infection, depression, a neurodegenerative disorder, trauma, age related cataracts, organ transplant rejection, or an autoimmune disease.;SOLUTION: The present invention provides IDO1 inhibitors of a formula I or pharmaceutically acceptable salts thereof (In the formula, X, L, n, m, R1, R2a, R2b, Rn, Rm, and Rt each represent a specific atom, bond, repetition number, substituent or the like).;SELECTED DRAWING: None;COPYRIGHT: (C)2019,JPO&INPIT
机译:解决的问题:提供吲哚胺2,3-二加氧酶1(IDO1)抑制剂,用于治疗癌症,病毒感染,抑郁症,神经退行性疾病,创伤,与年龄有关的白内障,器官移植排斥或自身免疫性疾病。本发明提供式I的IDO1抑制剂或其药学上可接受的盐(在式中,X,L,n,m,R 1 ,R 2a ,R 2b ,R n ,R m 和R t 分别表示特定的原子,键,重复数,取代基或;选择的图纸:无;版权:(C)2019,JPO&INPIT

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