embedded image ;wherein custom-character is a single or double bond, X is NCH3 or CH2, Y is null, O or N, R1 is H, OH, and R2 is null, H, C1-C8 alkyl, —(C═O)-alkyl, —(C═O)-aryl, —(C═O)-alkyl-aryl, —(C═O)-heteroaryl, cycloalkyl or heterocycloalkyl, which optionally substituted by one or more of —OH, —NO2, —NH2, —NR3R4, carbonyl, alkoxyl, alkyl or —OCF3, wherein R3 and R4 independently are H, alkyl, —SO2CH3, —(C═O)—CH3 or —(C═O)—NH2."/> METHOD FOR TREATING AN AUTOIMMUNE NEUROLOGICAL DISEASE AND/OR NEURODEGENERATIVE DISEASE AND PHARMACEUTICAL FORMULATIONS FOR A LIQUID DOSAGE FORM AND A CONTROLLED RELEASE DOSAGE FORM
首页> 外国专利> METHOD FOR TREATING AN AUTOIMMUNE NEUROLOGICAL DISEASE AND/OR NEURODEGENERATIVE DISEASE AND PHARMACEUTICAL FORMULATIONS FOR A LIQUID DOSAGE FORM AND A CONTROLLED RELEASE DOSAGE FORM

METHOD FOR TREATING AN AUTOIMMUNE NEUROLOGICAL DISEASE AND/OR NEURODEGENERATIVE DISEASE AND PHARMACEUTICAL FORMULATIONS FOR A LIQUID DOSAGE FORM AND A CONTROLLED RELEASE DOSAGE FORM

机译:治疗液体剂量形式和控制释放剂量形式的自发性神经疾病和/或神经退行性疾病和药物制剂的方法

摘要

A method for treating an autoimmune neurological disease and/or a neurodegenerative disease is provided. The method includes administering an effective amount of at least one compound having Formula (I), Formula (II) or Formula (III), or its geometric isomer, enantiomer or diastereomer to a subject in need thereof:; embedded image ;wherein custom-character is a single or double bond, X is NCH3 or CH2, Y is null, O or N, R1 is H, OH, and R2 is null, H, C1-C8 alkyl, —(C═O)-alkyl, —(C═O)-aryl, —(C═O)-alkyl-aryl, —(C═O)-heteroaryl, cycloalkyl or heterocycloalkyl, which optionally substituted by one or more of —OH, —NO2, —NH2, —NR3R4, carbonyl, alkoxyl, alkyl or —OCF3, wherein R3 and R4 independently are H, alkyl, —SO2CH3, —(C═O)—CH3 or —(C═O)—NH2.
机译:提供了一种用于治疗自身免疫性神经疾病和/或神经变性疾病的方法。该方法包括将有效量的至少一种具有式(I),式(II)或式(III)的化合物或其几何异构体,对映异构体或非对映异构体给予需要其的受试者: “嵌入式图像” ;其中“是单个或双键,X为NCH 3 或CH 2 ,Y为零,O或N,R 1 为H,OH和R < Sub> 2 为空,H,C 1 -C 8 烷基,-(C═O)-烷基,-(C═O)-芳基,-(C═O)-烷基-芳基,-(C═O)-杂芳基,环烷基或杂环烷基,它们任选被-OH,-NO 2 ,-NH < Sub> 2 ,-NR 3 R 4 ,羰基,烷氧基,烷基或-OCF 3 ,其中R 3 和R 4 独立地是H,烷基,-SO 2 CH 3 ,-(C═O)-CH < Sub> 3 或-(C═O)-NH 2

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