首页> 外国专利> METHOD FOR TREATING AN AUTOIMMUNE NEUROLOGICAL DISEASE AND/OR NEURODEGENERATIVE DISEASE AND PHARMACEUTICAL FORMULATIONS FOR A LIQUID DOSAGE FORM AND A CONTROLLED RELEASE DOSAGE FORM

METHOD FOR TREATING AN AUTOIMMUNE NEUROLOGICAL DISEASE AND/OR NEURODEGENERATIVE DISEASE AND PHARMACEUTICAL FORMULATIONS FOR A LIQUID DOSAGE FORM AND A CONTROLLED RELEASE DOSAGE FORM

机译:治疗液体剂量形式和控制释放剂量形式的自发性神经疾病和/或神经退行性疾病和药物制剂的方法

摘要

wherein is a single or double bond, X is NCH3 or CH2, Y is null, O or N, R1 is H, OH, and R2 is null, H, C1-C8 alkyl, —(C═O)-alkyl, —(C═O)-aryl, —(C═O)-alkyl-aryl, —(C═O)-heteroaryl, cycloalkyl or heterocycloalkyl, which optionally substituted by one or more of —OH, —NO2, —NH2, —NR3R4, carbonyl, alkoxyl, alkyl or —OCF3, wherein R3 and R4 independently are H, alkyl, —SO2CH3, —(C═O)—CH3 or —(C═O)—NH2.
机译:其中为单键或双键,X为NCH3或CH2,Y为零,O或N,R1为H,OH,R2为零,H,C1-C8烷基,-(C═O)-烷基,- (C═O)-芳基,-(C═O)-烷基-芳基,-(C═O)-杂芳基,环烷基或杂环烷基,其任选地被-OH,-NO2,-NH2,-中的一个或多个取代NR 3 R 4,羰基,烷氧基,烷基或-OCF 3,其中R 3和R 4独立地为H,烷基,-SO 2 CH 3,-(C = O)-CH 3或-(C = O)-NH 2。

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