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CRYSTALLIC FORMS OF LYSYLOXIDASE-LIKE PROTEIN 2 INHIBITOR AND METHODS FOR PRODUCING

机译:溶血脂酶样蛋白2抑制剂的结晶形式及其制备方法

摘要

This document describes the crystalline forms of the pharmaceutically acceptable salts of the lysyl oxidase-like protein 2 (LOXL2) (3- (4- (aminomethyl) -6- (trifluoromethyl) pyridin-2-yloxy) phenyl) ((3R, 4R) -3- fluoro-4-hydroxypyrrolidin-1-yl) methanone. Methods for preparing a LOXL2 inhibitor, pharmaceutical compositions and drugs containing a LOXL2 inhibitor, and methods for using a LOXL2 inhibitor in the treatment of conditions, diseases, or disorders associated with LOXL2 activity are also described.
机译:该文件描述了赖氨酰氧化酶样蛋白2(LOXL2)(3-(4-(氨基甲基)-6-(三氟甲基)吡啶-2-基氧基)苯基)((3R,4R )-3-氟-4-羟基吡咯烷-1-基)甲酮。还描述了制备LOXL2抑制剂的方法,包含LOXL2抑制剂的药物组合物和药物,以及在治疗与LOXL2活性有关的状况,疾病或病症中使用LOXL2抑制剂的方法。

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