首页> 外国专利> PHTHALAZINE DERIVATIVES AS INHIBITORS OF PARP1, PARP2 AND/OR TUBULIN USEFUL FOR THE TREATMENT OF CANCER.

PHTHALAZINE DERIVATIVES AS INHIBITORS OF PARP1, PARP2 AND/OR TUBULIN USEFUL FOR THE TREATMENT OF CANCER.

机译:酞嗪衍生物可作为PARP1,PARP2和/或微管蛋白的抑制剂,可用于治疗癌症。

摘要

The application relates to phthalazine derivatives of formula (I) which are inhibitors of PARP1, PARP2 and/or tubulin and thus useful for the treatment of cancer. Also disclosed are pharmaceutical formulations containing such compounds, as well as combinations of these compounds with at least one additional therapeutic agent.
机译:本申请涉及式(I)的酞嗪衍生物,其是PARP1,PARP2和/或微管蛋白的抑制剂,因此可用于治疗癌症。还公开了包含此类化合物的药物制剂,以及这些化合物与至少一种其他治疗剂的组合。

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