首页> 外国专利> PYRAZOLES DERIVATIVES MODULATORS OF CALCIUM RELEASE-ACTIVATED CALCIUM CHANNEL AND METHODS FOR TREATMENT OF NON-SMALL CELL LUNG CANCER

PYRAZOLES DERIVATIVES MODULATORS OF CALCIUM RELEASE-ACTIVATED CALCIUM CHANNEL AND METHODS FOR TREATMENT OF NON-SMALL CELL LUNG CANCER

机译:钙释放活化钙通道的吡咯衍生物调节剂及非小细胞肺癌的治疗方法

摘要

Dislcosed are novel calcium release-activated calcium (CRAC) channelinhibitors, such as(see above formula), methods for preparing them, pharmaceuticalcompositions containing them, and methods of treatment using them. The presentdislcosurealso relates to methods for treating non-small cell lung cancer (NSCLC) withCRACinhibitors, and to methods for identifying therapeutics for treating and ofdiagnosing cancer.
机译:揭示了新的钙释放激活钙(CRAC)通道抑制剂,例如(请参见上式),制备方法,药物含有它们的组合物,以及使用它们的治疗方法。现在揭露还涉及治疗非小细胞肺癌(NSCLC)的方法CRAC抑制剂,以及鉴定用于治疗和治疗的疗法的方法诊断癌症。

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